Efficient and regiospecific one-pot synthesis of substituted 1,2,4-triazoles

被引：77
|
作者：
Stocks, MJ [1 ]
Cheshire, DR [1 ]
Reynolds, R [1 ]
机构：
[1] AstraZeneca R&D Charnwood, Dept Med Chem, Loughborough LE11 5RH, Leics, England
来源：
ORGANIC LETTERS | 2004年 / 6卷 / 17期
关键词：
D O I：
10.1021/ol048863a
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient one-pot, three-component synthesis of substituted 1,2,4-triazoles has been developed, utilizing a wide range of substituted primary amines and acyl hydrazides.
引用
收藏
页码：2969 / 2971
页数：3
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