Rapid optimization of LFA-1/ICAM-1 and Mac-1/ICAM-1 antagonists via a parallel synthesis approach.

被引:0
|
作者
Yun, WY [1 ]
Desai, BB [1 ]
Du, Y [1 ]
Fotouhi, N [1 ]
Gillespie, P [1 ]
Guthrie, RW [1 ]
Huang, KS [1 ]
Kolinsky, K [1 ]
Li, SH [1 ]
Mennona, FA [1 ]
Perrotta, A [1 ]
Pietranico-Cole, SL [1 ]
Portland, L [1 ]
Vermeulen, J [1 ]
机构
[1] Hoffmann La Roche Inc, Roche Res Ctr, Nutley, NJ 07110 USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
321-MEDI
引用
收藏
页码:U63 / U63
页数:1
相关论文
共 50 条
  • [1] LFA-1 mediates neutrophil transendothelial migration via engagement of ICAM-1 and ICAM-2, but Mac-1 mediated migration is not ICAM-1 or -2 dependent.
    Issekutz, AC
    Springer, TA
    [J]. JOURNAL OF ALLERGY AND CLINICAL IMMUNOLOGY, 1997, 99 (01) : 482 - 482
  • [2] Role of LFA-1 and ICAM-1 in Cancer
    Reina, Manuel
    Espel, Enric
    [J]. CANCERS, 2017, 9 (11):
  • [3] Elucidating the kinetics of LFA-1 and Mac-1 sequential binding to ICAM-1 under shear conditions
    Eniola, AO
    Smith, CW
    [J]. FASEB JOURNAL, 2006, 20 (05): : A1080 - A1081
  • [4] Activated polymorphonuclear leukocytes induce constriction of canine coronary artery via Mac-1, but not LFA-1, and ICAM-1
    Minamino, T
    Kitakaze, M
    Node, K
    Funaya, H
    Inoue, M
    Hori, M
    Kamada, T
    [J]. JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 1996, 28 (07) : 1575 - 1581
  • [5] Practical synthesis of LFA-1/ICAM-1 inhibitors.
    Farina, V
    Napolitano, E
    Eriksson, M
    Kapadia, S
    Spero, D
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 222 : U69 - U69
  • [6] LFA-1 AND ICAM-1 IN LYMPHOCYTE-ACTIVATION
    BRANDEN, H
    HEDMAN, H
    LUNDGREN, E
    [J]. SCANDINAVIAN JOURNAL OF IMMUNOLOGY, 1990, 32 (04) : 386 - 386
  • [7] MEASUREMENT OF THE AFFINITY OF THE ICAM-1/LFA-1 INTERACTION
    LOLLO, BA
    MOY, VT
    BRIAN, AA
    [J]. FASEB JOURNAL, 1991, 5 (05): : A996 - A996
  • [8] Expression and significance of ICAM-1 and its counter receptors LFA-1 and Mac-1 in experimental acute pancreatitis of rats
    Yasuhiro Watanabe
    [J]. World Journal of Gastroenterology, 2006, (31) : 5005 - 5009
  • [9] Synergistic inhibitory activity of α- and β-LFA-1 peptides on LFA-1/ICAM-1 interaction
    Yusuf-Makagiansar, H
    Makagiansar, IT
    Hu, YB
    Siahaan, TJ
    [J]. PEPTIDES, 2001, 22 (12) : 1955 - 1962
  • [10] Expression and significance of ICAM-1 and its counter receptors LFA-1 and Mac-1 in experimental acute pancreatitis of rats
    Sun, Wei
    Watanabe, Yasuhiro
    Wang, Zhong-Qiu
    [J]. WORLD JOURNAL OF GASTROENTEROLOGY, 2006, 12 (31) : 5005 - 5009