New access to thiazolo[4,5-d]pyrimidine derivatives

被引：41

作者：

Bakavoli, M. ^{[1
]}

Nikpour, M. ^{[1
]}

Rahimizadeh, M. ^{[1
]}

机构：

[1] Ferdowsi Univ Mashhad, Sch Sci, Dept Chem, Mashhad 917751436, Iran

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2006年 / 43卷 / 05期

关键词：

D O I：

10.1002/jhet.5570430527

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

4-Amino-5-bromo-2-substituted-aminopyrimidines are readily obtained from the newly prepared 5-bromo-2,4-dichloro-6-methylpyrimidine by sequential treatment with ethanolic ammonia and secondary amines. These compounds were successfully reacted with various isothiocyanates in the presence of sodamide in DMF to form the new thiazolo[4,5-d] pyrimidine derivatives.

引用

页码：1327 / 1329

页数：3

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