Facile synthesis of a selectively protected triazamacrocycle

被引：4
|
作者：
Skerlj, RT [1 ]
Nan, SQ [1 ]
Zhou, YX [1 ]
Bridger, GJ [1 ]
机构：
[1] AnorMED Inc, Langley, BC V2Y 1N5, Canada
来源：
TETRAHEDRON LETTERS | 2002年 / 43卷 / 42期
关键词：
D O I：
10.1016/S0040-4039(02)01756-2
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
1,7-Diaminoheptane was selectively homologated with the novel reagent N-(2-nitrobenzenesulfonyl)aziridine. A series of reactions then followed to afford a selectively protected 14-membered triazamacrocyclic ring. (C) 2002 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：7569 / 7571
页数：3
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