SYNTHESIS OF NOVEL FAC-[99MTc(CO)3+]-LABELED (±)-NICOTINE AND A-84543 ANALOGS AS POTENTIAL α4β2 NEURONAL NICOTINIC RECEPTOR IMAGING AGENTS

被引：0

作者：

Papagiannopoulou, D. ^{[1
]}

Kramer, D. J. ^{[2
]}

Mamhood, A. ^{[1
]}

Davison, A. ^{[2
]}

Jones, A. G. ^{[1
]}

机构：

[1] Harvard Univ, Sch Med, Boston, MA USA

[2] MIT, Cambridge, MA 02139 USA

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2005年 / 48卷

关键词：

Technetium; Nicotinic Acetylcholine Receptors; Tc(CO)(3) Complexes;

D O I：

暂无

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

引用

页码：S245 / S245

页数：1

共 49 条

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[45] Versatile synthetic approach to new bifunctional chelating agents tailor made for labeling with the fac-[M(CO)3]+ core (M = Tc, 99mTc, Re):: synthesis, in vitro, and in vivo behavior of the model complex [M(APPA)(CO)3] (APPA = [(5-amino-pentyl)-pyridin-2-yl-methyl-amino]-acetic acid)
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[48] Synthesis, characterization and X-ray crystal structure of [Re(L4)(CO)3]Br • 2CH3OH (L4=N,N-bis[(2-diphenylphosphino)ethyl]-methoxyethylamine):: A model compound for novel cationic 99mTc(I)-tricarbonyl radiotracers useful for heart imaging
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