An Improved Process for the Synthesis of 4H-Imidazo[1,5-a][1,4]benzodiazepines

被引：11
|
作者：
Yang, Jie [1 ]
Teng, Yun [1 ]
Ara, Shamim [1 ]
Rallapalli, Sundari [1 ]
Cook, James M. [1 ]
机构：
[1] Univ Wisconsin, Dept Chem, Milwaukee, WI 53211 USA
来源：
SYNTHESIS-STUTTGART | 2009年 / 06期
关键词：
GABA(A)/Bz receptors; imidazo[1,5-a][1,4]benzodiazepines; ethyl isocyanoacetate; annulation; BENZODIAZEPINE; IMIDAZOBENZODIAZEPINES; PHARMACOPHORE; SUBSTITUENTS; SUBTYPES; LIGANDS; PROBES;
D O I：
10.1055/s-0028-1083358
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The construction of CNS active imidazo[1,5-a][1,4]benzodiazepines has been improved in a one-pot annulation process.
引用
收藏
页码：1036 / 1040
页数：5
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