Novel 3,5-diaryl pyrazolines as human acyl-CoA:cholesterol acyltransferase inhibitors (vol 14, pg 3109, 2004)

被引：0

作者：

Jeong, Tae-Sook ^{[1
]}

Kim, Kyung Soon ^{[1
]}

An, Sojin ^{[1
]}

Cho, Kyung-Hyun ^{[1
]}

Lee, Sangku ^{[1
]}

Lee, Woo Song ^{[1
]}

机构：

[1] Korea Res Inst Biosci & Biotechnol, Natl Res Lab Lipid Metab & Atherosclerosis, Taejon 305333, South Korea

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 2009年 / 19卷 / 08期

关键词：

D O I：

10.1016/j.bmcl.2004.03.113

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：2364 / 2364

页数：1

共 47 条

[41] Synthesis and biological activity of novel 4-phenyl-1,8-naphthyridin-2(1H)-on-3-yl ureas:: Potent acyl-CoA:cholesterol acyltransferase inhibitor with improved aqueous solubility
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BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (01) : 44 - 48
[42] Human acyl-coenzyme A: Cholesterol acyltransferase 2 (hACAT2) expressed in Chinese hamster ovary cells: Membrane topology and active site location (vol 14, pg 2447, 2003)
Lin, S
Lu, S
Chang, CCY
Chang, TY
MOLECULAR BIOLOGY OF THE CELL, 2003, 14 (10)
[43] The metabolic stability of acyl-CoA:cholesterol O-acyltransferase (ACAT) inhibitors, N-(4-benzyloxy-3,5-dimethoxycinnamoyl)-N′-(2,4-dimethylphenyl)piperazine (YIC-708-424) and its derivatives in rat liver and intestinal epithelium
Ohishi, K
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Hatano, H
Aiyama, R
Watanabe, T
Yokokura, T
BIOLOGICAL & PHARMACEUTICAL BULLETIN, 2003, 26 (05) : 600 - 607
[44] 2,3,22,23-Tetrahydroxyl-2,6,10,15,19,23-hexamethyl-6,10,14,18-tetracosatetraene, an Acyclic Triterpenoid Isolated from the Seeds of Alpinia katsumadai, Inhibits Acyl-CoA: Cholesterol Acyltransferase Activity
Choi, Soon-Yong
Lee, Moon Hee
Choi, Jung Ho
Kim, Young Kook
BIOLOGICAL & PHARMACEUTICAL BULLETIN, 2012, 35 (11) : 2092 - 2096
[45] 1-(2,6-diisopropylphenyl)-3-(1,3-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8/7-ylalkyl)ureas as potential acyl-CoA:cholesterol acyltransferase inhibitors
Rybár, A
Alföldi, J
Faberová, V
Schmidtová, L'
CHEMICAL PAPERS-CHEMICKE ZVESTI, 2002, 56 (05): : 330 - 339
[46] STRUCTURE-ACTIVITY RELATIONSHIP OF N-[2-(DIMETHYLAMINO)-6-[3-(5-METHYL-4-PHENYL-1H-IMIDAZOL-1-YL)PROPOXY]PHENYL]-N'-PENTYLUREA AND ANALOGS - NOVEL POTENT INHIBITORS OF ACYL-COA CHOLESTEROL O-ACYLTRANSFERASE WITH ANTIATHEROSCLEROTIC ACTIVITY
KIMURA, T
TAKASE, Y
HAYASHI, K
TANAKA, H
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SAEKI, T
KOGUSHI, M
YAMADA, T
FUJIMORI, T
SAITOU, I
AKASAKA, K
JOURNAL OF MEDICINAL CHEMISTRY, 1993, 36 (11) : 1630 - 1640
[47] SYNTHESES AND PHARMACOLOGICAL ACTIVITIES OF NOVEL OPTICALLY-ACTIVE INHIBITORS OF ACYL-COA - CHOLESTEROL O-ACYLTRANSFERASE - EAB-309 ((R)-N-2-(1,3-BENZODIOXOL-4-YL)HEPTYL-N'-2,6-DIISOPROPYLPHENYLUREA) AND ITS ENANTIOMER
SEKIYA, T
INOUE, S
SHIRASAKA, T
MIYAJIMA, C
OKUSHIMA, H
SUZUKI, K
KAWAI, M
MITSUKA, M
UMEZU, K
CHEMICAL & PHARMACEUTICAL BULLETIN, 1994, 42 (03) : 586 - 591

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