In vitro discrimination between sedative and non-sedative histamine H1 receptor antagonists by an intact cell binding assay.

被引：0
|
作者：
Shigeru, Hishinuma
Masaki, Saito
机构：
来源：
ACTA PHARMACOLOGICA SINICA | 2006年 / 27卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
引用
收藏
页码：360 / 360
页数：1
相关论文
共 37 条
  • [21] Inhibitory action of histamine H1 receptor antagonists on eosinophil functions in vitro and in vivo
    Furuta, A.
    Kanai, K.
    Asano, K.
    Suzaki, H.
    Suzuki, M.
    ALLERGY, 2010, 65 : 519 - 519
  • [22] Interactions between histamine H1 receptor and its antagonists by using cell membrane chromatography method
    Ma, Weina
    Zhang, Dongdong
    Li, Jing
    Che, Delu
    Liu, Rui
    Zhang, Jie
    Zhang, Yanmin
    JOURNAL OF PHARMACY AND PHARMACOLOGY, 2015, 67 (11) : 1567 - 1574
  • [23] PET measurement of brain histamine H1 receptor occupancy of an orally-administered antihistamine, bepotastine, and its sedative property
    Tashiro, M.
    Duan, X.
    Kato, M.
    Iwata, R.
    Itoh, M.
    Yanai, K.
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2008, 35 : S130 - S131
  • [24] In vitro inhibition of CYP3A4 by histamine H1 receptor antagonists.
    Hamelin, BA
    Gauvin, C
    Turgeon, J
    CLINICAL PHARMACOLOGY & THERAPEUTICS, 1997, 61 (02) : PIV30 - PIV30
  • [25] Potential central sedative effect of antihistamine eye-drops: histamine H1 receptor occupancy measured by positron emission tomography
    Zhang, Dongying
    Shibuya, Katsuhiko
    Tashiro, Manabu
    Harada, Ryuichi
    Okamura, Nobuyuki
    Yoshikawa, Takeo
    Yanai, Kazuhiko
    JOURNAL OF PHARMACOLOGICAL SCIENCES, 2011, 115 : 221P - 221P
  • [26] Suppressive activity of histamine H1 receptor antagonists, desloratadine and levocetirizine, on the production of periostin in vitro.
    Asano, M.
    Mizuyoshi, T.
    Furuta, A.
    Asano, K.
    Kobayashi, H.
    ALLERGY, 2017, 72 : 290 - 290
  • [27] H-1 BUT NOT H-2-HISTAMINE RECEPTOR ANTAGONISTS PRODUCE CEREBRAL ARTERIOLAR CONSTRICTION - POSSIBLE EXPLANATION OF THE SEDATIVE AND SOPORIFIC EFFECTS OF ANTIHISTAMINES
    LASSOFF, S
    ALTURA, BM
    FEDERATION PROCEEDINGS, 1983, 42 (03) : 486 - 486
  • [28] EVALUATION OF RESIDUAL SEDATIVE EFFECT OF ANTIHISTAMINES BY MEASURING CENTRAL HISTAMINE H1 RECEPTOR OCCUPANCY USING 11C-DOXEPIN-PET
    Yanai, Kazuhiko
    Zhang, Dongying
    Manabu, Tashiro
    Shibuya, Katsuhiko
    ACTA DERMATO-VENEREOLOGICA, 2009, 89 (06) : 707 - 707
  • [29] Characterization of interactions between local anesthetics and histamine H1 receptor by cell membrane chromatography model
    Cao, Jiao
    Yang, Liu
    Wang, Yuejin
    Liu, Rui
    Zhang, Tao
    He, Langchong
    JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2021, 196
  • [30] In vitro characterization of cytochrome P450 2D6 inhibition by classic histamine H1 receptor antagonists
    Hamelin, BA
    Bouayad, A
    Drolet, B
    Gravel, A
    Turgeon, J
    DRUG METABOLISM AND DISPOSITION, 1998, 26 (06) : 536 - 539
1234