Annellation of triazole and tetrazole systems onto pyrrolo[2,3-d]pyrimidines:: Synthesis of tetrazolo[1,5-c]pyrrolo[3,2-e]-pyrimidines and triazolo[1,5-c]pyrrolo-[3,2-e]pyrimidines as potential antibacterial agents

被引：39

作者：

Dave, CG ^{[1
]}

Shah, RD ^{[1
]}

机构：

[1] MG Sci Inst, Organ Synth Lab, Ahmedabad 380009, Gujarat, India

来源：

MOLECULES | 2002年 / 7卷 / 07期

关键词：

tetrazolopyrrolopyrimidines; triazolopyrrolopyrimidines; pyrrolo[2,3-d]pyrimidines; antibacterial activity;

D O I：

10.3390/70700554

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

Syntheses of several novel 4-chloropyrrolo[2,3-d]pyrimidines (1), 4-hydrazinopyrrolo[2,3-d]pyrimidines (2) and 3-amino-4-iminopyrrolo[2,3-d]pyrimidines (7) and their use in the synthesis of tetrazolo[1,5-c]pyrrolo[3,2-e]pyrimidines (3) and triazolo[1,5-c]pyrrolo[3,2-e]pyrimidines (4) required for biological screening are reported.

引用

页码：554 / 565

页数：12

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