Annellation of triazole and tetrazole systems onto pyrrolo[2,3-d]pyrimidines:: Synthesis of tetrazolo[1,5-c]pyrrolo[3,2-e]-pyrimidines and triazolo[1,5-c]pyrrolo-[3,2-e]pyrimidines as potential antibacterial agents

被引：39

作者：

Dave, CG ^{[1
]}

Shah, RD ^{[1
]}

机构：

[1] MG Sci Inst, Organ Synth Lab, Ahmedabad 380009, Gujarat, India

来源：

MOLECULES | 2002年 / 7卷 / 07期

关键词：

tetrazolopyrrolopyrimidines; triazolopyrrolopyrimidines; pyrrolo[2,3-d]pyrimidines; antibacterial activity;

D O I：

10.3390/70700554

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

Syntheses of several novel 4-chloropyrrolo[2,3-d]pyrimidines (1), 4-hydrazinopyrrolo[2,3-d]pyrimidines (2) and 3-amino-4-iminopyrrolo[2,3-d]pyrimidines (7) and their use in the synthesis of tetrazolo[1,5-c]pyrrolo[3,2-e]pyrimidines (3) and triazolo[1,5-c]pyrrolo[3,2-e]pyrimidines (4) required for biological screening are reported.

引用

页码：554 / 565

页数：12

共 50 条

[1] Synthesis of fused tetrazolo[1,5-c] pyrrolo[3,2-e]pyrimidines and their reductive conversion to new 4-aminopyrrolo[2,3-d]pyrimidines
Desai, Nirmal D.
SYNTHETIC COMMUNICATIONS, 2006, 36 (15) : 2169 - 2182
[2] Synthesis of 7H-tetrazolo[1,5-c]pyrrolo[3,2-e]pyrimidines and their reductive ring cleavage to 4-aminopyrrolo[2,3-d]pyrimidines
Dave, CG
Shah, RD
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1998, 35 (06) : 1295 - 1300
[3] DMAP catalyzed synthesis of some new pyrrolo[3,2-e][1,2,4]triazolo[1,5-c]pyrimidines
Khashi, Maryam
Davoodnia, Abolghasem
Lingam, V. S. Prasada Rao
RESEARCH ON CHEMICAL INTERMEDIATES, 2015, 41 (08) : 5731 - 5742
[4] DMAP catalyzed synthesis of some new pyrrolo[3,2-e][1,2,4]triazolo[1,5-c]pyrimidines
Maryam Khashi
Abolghasem Davoodnia
V. S. Prasada Rao Lingam
Research on Chemical Intermediates, 2015, 41 : 5731 - 5742
[5] Synthesis of substituted furo[3,2-e][1,2,4]triazolo[4,3-c]pyrimidines and furo[3,2-e]tetrazolo[1,5-c]pyrimidines
Lockhart, CC
Sowell, JW
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1996, 33 (03) : 659 - 661
[6] Synthesis of substituted furo[3,2-e][1,2,4]triazolo[4,3-c]pyrimidines and furo[3,2-e]tetrazolo[1,5-c]pyrimidines.
Lockhart, CC
Sowell, JW
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1996, 211 : 235 - ORGN
[7] SYNTHESIS AND BIOLOGICAL-ACTIVITY OF TETRAZOLO[1,5-C]THIENO[3,2-E]PYRIMIDINES
SHISHOO, CJ
DEVANI, MB
KARVEKAR, MD
ULLAS, GV
ANANTHAN, S
BHADTI, VS
PATEL, RB
GANDHI, TP
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1982, 21 (07): : 666 - 668
[8] Synthesis of new furo[2,3-d]pyrimidines and furo[3,2-e][1,2,4]triazolo[1,5-c]pyrimidines
Shaker, Raafat M.
ARKIVOC, 2006, : 68 - 77
[9] Synthesis and rearrangements of 7H-pyrrolo[3,2-e][1,2,4]triazolo[1,5-c]and 7H-pyrrolo[3,2-e][1,2,4]triazolo[4,3-c]pyrimidines
Vorob'ev, E. V.
Kurbatov, E. S.
Krasnikov, V. V.
Mezheritskii, V. V.
Usova, E. V.
RUSSIAN CHEMICAL BULLETIN, 2006, 55 (08) : 1492 - 1497
[10] Synthesis and rearrangements of 7H-pyrrolo[3,2-e][1,2,4]triazolo[1,5-c]-and 7h-pyrrolo[3,2-e][1,2,4]triazolo[4,3-c]pyrimidines
E. V. Vorob’ev
E. S. Kurbatov
V. V. Krasnikov
V. V. Mezheritskii
E. V. Usova
Russian Chemical Bulletin, 2006, 55 : 1492 - 1497

← 1 2 3 4 5 →