An Allosteric Region of Src Tyrosine Kinase Allows for Stabilization of Its Active-Like Conformation

被引:0
|
作者
Ahuja, Lalima G. [1 ]
Meng, Yilin [2 ]
Kornev, Alexandr P. [3 ]
Roux, Benoit [2 ]
Taylor, Susan [4 ]
机构
[1] Univ Calif San Diego, Pharmacol, San Deigo, CA USA
[2] Univ Chicago, Biochem & Mol Biol, Chicago, IL 60637 USA
[3] Univ Calif San Diego, Pharmacol, San Diego, CA 92103 USA
[4] Univ Calif San Diego, Pharmacol, Chem Biochem, San Diego, CA 92103 USA
关键词
D O I
10.1016/j.bpj.2017.11.2201
中图分类号
Q6 [生物物理学];
学科分类号
071011 ;
摘要
1959-Plat
引用
收藏
页码:398A / 398A
页数:1
相关论文
共 50 条
  • [31] Ixodes scapularis Src tyrosine kinase facilitates Anaplasma phagocytophilum survival in its arthropod vector
    Turck, Jeremy W.
    Taank, Vikas
    Neelakanta, Girish
    Sultana, Hameeda
    TICKS AND TICK-BORNE DISEASES, 2019, 10 (04) : 838 - 847
  • [32] CLONING OF FRK, A NOVEL HUMAN INTRACELLULAR SRC-LIKE TYROSINE KINASE-ENCODING GENE
    LEE, J
    WANG, ZY
    LUOH, SM
    WOOD, WI
    SCADDEN, DT
    GENE, 1994, 138 (1-2) : 247 - 251
  • [33] The positive allosteric modulator BPAM344 and L-glutamate introduce an active-like structure of the ligand-binding domain of GluK2
    Bay, Yasmin
    Jeppesen, Mie Egeberg
    Frydenvang, Karla
    Francotte, Pierre
    Pirotte, Bernard
    Pickering, Darryl S.
    Kristensen, Anders Skov
    Kastrup, Jette Sandholm
    FEBS LETTERS, 2024, 598 (07) : 743 - 757
  • [34] Tamoxifen-resistant variants that are not killed by fulvestrant overexpress active c-Src tyrosine kinase.
    Planas-Silva, M. D.
    Hamilton, K., V
    BREAST CANCER RESEARCH AND TREATMENT, 2006, 100 : S194 - S194
  • [35] BACTERIAL EXPRESSION OF AN ACTIVE TYROSINE KINASE FROM A PROTEIN-A TRUNCATED C-SRC FUSION PROTEIN
    SAYA, H
    LEE, PSY
    NISHI, T
    IZAWA, I
    NAKAJIMA, M
    GALLICK, GE
    LEVIN, VA
    FEBS LETTERS, 1993, 327 (02) : 224 - 230
  • [36] ANTIBODIES TO A DEFINED REGION OF PP60SRC NEUTRALIZE THE TYROSINE-SPECIFIC KINASE-ACTIVITY
    GENTRY, LE
    ROHRSCHNEIDER, LR
    CASNELLIE, JE
    KREBS, EG
    JOURNAL OF BIOLOGICAL CHEMISTRY, 1983, 258 (18) : 1219 - 1228
  • [37] QUANTITATION OF A SRC-LIKE TYROSINE PROTEIN-KINASE DURING FERTILIZATION OF THE SEA-URCHIN EGG
    KAMEL, C
    VENO, PA
    KINSEY, WH
    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1986, 138 (01) : 349 - 355
  • [38] Src tyrosine kinase signaling antagonizes nuclear localization of FOXO and inhibits its transcription factor activity
    Buelow, Margret H.
    Buelow, Torsten R.
    Hoch, Michael
    Pankratz, Michael J.
    Juenger, Martin A.
    SCIENTIFIC REPORTS, 2014, 4
  • [39] Deregulation of c-Src tyrosine kinase and its downstream targets in pre-eclamptic placenta
    Irtegun, Sevgi
    Akcora-Yildiz, Dilara
    Pektanc, Gulsum
    Karabulut, Cagla
    JOURNAL OF OBSTETRICS AND GYNAECOLOGY RESEARCH, 2017, 43 (08) : 1278 - 1284
  • [40] The protein tyrosine kinase Src and its role upon alpha-toxin stimulation of human platelets
    Vogel, K.
    Burke, M.
    Presek, P.
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2012, 385 : 99 - 100