EZH2 inhibitors in immunotherapy of melanoma

被引：1
|
作者：
Hersey, Peter
Gallagher, Stuart
Tiffen, Jessamy
Shklovskaya, Elena
Wilson, Stephen
Filipp, Fabian
机构：
来源：
CANCER RESEARCH | 2017年 / 77卷
基金：
美国国家卫生研究院; 澳大利亚国家健康与医学研究理事会;
关键词：
D O I：
10.1158/1538-7445.AM2017-1676
中图分类号：
R73 [肿瘤学];
学科分类号：
100214 ;
摘要：
1676
引用
收藏
页数：2
相关论文
共 50 条
  • [31] EZH2 Inhibitors: Take It EZy, It Is All About Context
    Velcheti, Vamsidhar
    Wong, Kwok-Kin
    Saunthararajah, Yogen
    CANCER DISCOVERY, 2019, 9 (04) : 472 - 475
  • [32] Development of secondary mutations in wild-type and mutant EZH2 alleles cooperates to confer resistance to EZH2 inhibitors
    Gibaja, V.
    Shen, F.
    Harari, J.
    Korn, J.
    Ruddy, D.
    Saenz-Vash, V.
    Zhai, H.
    Rejtar, T.
    Paris, C. G.
    Yu, Z.
    Lira, M.
    King, D.
    Qi, W.
    Keen, N.
    Hassan, A. Q.
    Chan, H. M.
    ONCOGENE, 2016, 35 (05) : 558 - 566
  • [33] Biological evaluation of tanshindiols as EZH2 histone methyltransferase inhibitors
    Woo, Jimin
    Kim, Hyun-Young
    Byun, Byung Jin
    Chae, Chong-Hak
    Lee, Ji Young
    Ryu, Shi Yong
    Park, Woo-Kyu
    Cho, Heeyeong
    Choi, Gildon
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (11) : 2486 - 2492
  • [34] BET and EZH2 Inhibitors: Novel Approaches for Targeting Cancer
    Sofia Genta
    Maria Cristina Pirosa
    Anastasios Stathis
    Current Oncology Reports, 2019, 21
  • [35] The pleiotropic roles of EZH2 in T-cell immunity and immunotherapy
    Ying Wang
    Tien Bui
    Yi Zhang
    International Journal of Hematology, 2022, 116 : 837 - 845
  • [36] A patent review of EZH2 inhibitors from 2017 and beyond
    Wan, Guoquan
    Feng, Huan
    Su, Chang
    Zhu, Yongxia
    Zhang, Lidan
    Zhang, Qiangsheng
    Yu, Luoting
    EXPERT OPINION ON THERAPEUTIC PATENTS, 2023, 33 (04) : 293 - 308
  • [37] EZH2 inhibitors: a patent review (2014-2016)
    Stazi, Giulia
    Zwergel, Clemens
    Mai, Antonello
    Valente, Sergio
    EXPERT OPINION ON THERAPEUTIC PATENTS, 2017, 27 (07) : 797 - 813
  • [38] Synthesis and methylation inhibitory activity of EZH2 methyltransferase inhibitors
    Zhang, Xiaopan
    Yao, Zhiyi
    Jingxi Huagong/Fine Chemicals, 2020, 37 (10): : 2083 - 2089
  • [39] The pleiotropic roles of EZH2 in T-cell immunity and immunotherapy
    Wang, Ying
    Bui, Tien
    Zhang, Yi
    INTERNATIONAL JOURNAL OF HEMATOLOGY, 2022, 116 (06) : 837 - 845
  • [40] Discovery of novel bicyclic pyridone derivatives as inhibitors of EZH2
    Marx, Marx
    Bobinski, Thomas
    Briere, David
    Christensen, James
    Galemmo, Robert
    Lee, Matthew
    Sudhakar, Niranjan
    Winkelman, Jeff
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 255
12345