A Combretastatin Analogue C12 Binds to Colchicine Site in Tubulin, Inhibits Spindle Microtubule Dynamics, Activates Mitotic Checkpoint and Induces Apoptosis in Cancer Cells

被引:0
|
作者
Kumari, Anuradha [1 ]
Srivastava, Shalini [1 ]
Prassanawar, Shweta Shyam [1 ]
Sisodiya, Shailendra [2 ]
Guchhait, Sankar K. [2 ]
Panda, Dulal [1 ]
机构
[1] Indian Inst Technol, Dept Biosci & Bioengn, Mumbai, Maharashtra, India
[2] Natl Inst Pharmaceut Educ & Res, Dept Med Chem, Mohali, Punjab, India
关键词
D O I
暂无
中图分类号
Q6 [生物物理学];
学科分类号
071011 ;
摘要
2053-Pos
引用
收藏
页码:415A / 415A
页数:1
相关论文
共 1 条
  • [1] CXI-benzo-84 reversibly binds to tubulin at colchicine site and induces apoptosis in cancer cells
    Rai, Ankit
    Gupta, Tilak Kumar
    Kini, Sudarshan
    Kunwar, Ambarish
    Surolia, Avadhesha
    Panda, Dulal
    BIOCHEMICAL PHARMACOLOGY, 2013, 86 (03) : 378 - 391