Synthesis and antifungal activity of some new 1-aryl/heteroaryl-4-methyl-1,2,4-triazolo [4,3-a] quinoxalines

被引：0
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作者：
Aggarwal, Ranjana [1 ]
Sumran, Garima
Kumar, Rajiv
Aggarwal, Ashok
Parkash, Vipin
机构：
[1] Kurukshetra Univ, Dept Chem, Kurukshetra 136119, Haryana, India
[2] Kurukshetra Univ, Dept Bot, Kurukshetra 136119, Haryana, India
来源：
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2006年 / 16卷 / 01期
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D O I：
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中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A simple and highly efficient synthesis of some 1-aryl/heteroaryl-4-methyl-1,2,4-triazolo [4,3-a] quinoxalines (3) by oxidative cyclization of arene carbaldehyde-3-methylquinoxalin-2-yl hydrazones (2) with iodobenzene diacetate (IBD) in dichloromethane is described. Some of the compounds were tested in vitro for their antifungal activity against Fusarium udum, Helminthosporium sp. and Aspergillus flavus.
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页码：1 / 4
页数：4
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