Synthesis and antifungal activity of some new 1-aryl/heteroaryl-4-methyl-1,2,4-triazolo [4,3-a] quinoxalines

被引：0

作者：

Aggarwal, Ranjana ^{[1
]}

Sumran, Garima

Kumar, Rajiv

Aggarwal, Ashok

Parkash, Vipin

机构：

[1] Kurukshetra Univ, Dept Chem, Kurukshetra 136119, Haryana, India

[2] Kurukshetra Univ, Dept Bot, Kurukshetra 136119, Haryana, India

来源：

INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2006年 / 16卷 / 01期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A simple and highly efficient synthesis of some 1-aryl/heteroaryl-4-methyl-1,2,4-triazolo [4,3-a] quinoxalines (3) by oxidative cyclization of arene carbaldehyde-3-methylquinoxalin-2-yl hydrazones (2) with iodobenzene diacetate (IBD) in dichloromethane is described. Some of the compounds were tested in vitro for their antifungal activity against Fusarium udum, Helminthosporium sp. and Aspergillus flavus.

引用

页码：1 / 4

页数：4

共 50 条

[1] Copper(II) chloride mediated synthesis and DNA photocleavage activity of 1-aryl/heteroaryl-4-substituted-1,2,4-triazolo[4,3-a]quinoxalines
Aggarwal, Ranjana
Sumran, Garima
Kumar, Virender
Mittal, Ashwani
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2011, 46 (12) : 6083 - 6088
[2] Hypervalent iodine mediated synthesis of 1-aryl/hetryl-1,2,4-triazolo[4,3-a] pyridines and 1-aryl/hetryl 5-methyl-1,2,4-triazolo[4,3-a]quinolines as antibacterial agents
Sadana, AK
Mirza, Y
Aneja, KR
Prakash, O
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2003, 38 (05) : 533 - 536
[3] Synthesis of some new quinoxalines and 1,2,4-triazolo[4,3-a]-quinoxalines for evaluation of in vitro antitumor and antimicrobial activities
El-Hawash, Soad A. M.
Habib, Nargues S.
Kassem, Mervat A.
ARCHIV DER PHARMAZIE, 2006, 339 (10) : 564 - 571
[4] Tricyclic heteroaromatic systems. 1,2,4-triazolo[4,3-a]quinoxalines and 1,2,4-triazino[4,3-a]quinoxalines: Synthesis and central benzodiazepine receptor activity
Colotta, V
Catarzi, D
Varano, F
Cecchi, L
Filacchioni, G
Galli, A
Costagli, C
ARCHIV DER PHARMAZIE, 1997, 330 (12) : 387 - 391
[5] Synthesis and pharmacological activity of 1,2,4-triazolo[4,3-a]quinolines
Savini, L
Chiasserini, L
Pellerano, C
Filippelli, W
Falcone, G
FARMACO, 2001, 56 (12): : 939 - 945
[6] Synthesis and antimicrobial testing of thiazolinyl-, thiazolidinonyl-quinoxalines and 1,2,4-triazolo[4,3-a]quinoxalines
Habib, NS
ElHawash, SA
PHARMAZIE, 1997, 52 (08): : 594 - 598
[7] Synthesis and antimicrobial activity of 1-aryl-4-methyl (1,2,4) triazolo (4,3,a) quinoxalines
Vyas, DA
Chauhan, NA
Parikh, AR
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2005, 14 (04) : 361 - 362
[8] SYNTHESIS OF (PYRIDINYL)-1,2,4-TRIAZOLO[4,3-A]PYRIDINES
MORAN, DB
MORTON, GO
ALBRIGHT, JD
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1986, 23 (04) : 1071 - 1077
[9] Quinoxaline derivatives part II: Synthesis and antimicrobial testing of 1,2,4-triazolo[4,3-a]quinoxalines, 1,2,4-triazino[4,3-a]quinoxalines and 2-pyrazolylquinoxalines
El-Hawash, SA
Habib, NS
Fanaki, NH
PHARMAZIE, 1999, 54 (11): : 808 - 813
[10] SYNTHESIS AND PHYSICOCHEMICAL STUDY OF 1,2,4-TRIAZOLO[4,3-A]PYRIDINES AND 1,2,4-TRIAZOLO[2,3-A]PYRIDINES
BOUTEAU, B
LANCELOT, JC
ROBBA, M
JOURNAL OF HETEROCYCLIC CHEMISTRY, 1990, 27 (06) : 1649 - 1651

← 1 2 3 4 5 →