Discovery of Selective Dual Inhibitors of Bromodomain Protein BRD4 and JAK2 for Treatment of Hematologic Malignancies

被引：1

作者：

Upadhayaya, Ram S. ^{[1
]}

Kethiri, Raghava Reddy ^{[1
]}

Vellanki, Avanish ^{[2
]}

Lightfoot, Jeff ^{[3
]}

Local, Andrea ^{[4
]}

Rice, William G. ^{[4
]}

机构：

[1] Laxai Avanti Life Sci, Hyderabad, Andhra Pradesh, India

[2] Aptose Biosci Inc, Redwood City, CA USA

[3] Aptose Biosci Inc, Mississauga, ON, Canada

[4] Aptose Biosci Inc, San Diego, CA USA

来源：

BLOOD | 2016年 / 128卷 / 22期

关键词：

D O I：

10.1182/blood.V128.22.5212.5212

中图分类号：

R5 [内科学];

学科分类号：

1002 ; 100201 ;

摘要：

5212

引用

页数：4

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