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- [1] Discovery of Novel PI3Kδ Inhibitors Based on the p110δ Crystal Structure[J]. MOLECULES, 2022, 27 (19):Jia, Wenqing论文数: 0 引用数: 0 h-index: 0机构: Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R China Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R ChinaLuo, Shuyu论文数: 0 引用数: 0 h-index: 0机构: Tianjin Med Univ, Hosp Stomatol, Sch Stomatol, Tianjin 300070, Peoples R China Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R ChinaZhao, Wennan论文数: 0 引用数: 0 h-index: 0机构: Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R China Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R ChinaXu, Weiren论文数: 0 引用数: 0 h-index: 0机构: Tianjin Inst Pharmaceut Res, Tianjin 300070, Peoples R China Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R ChinaZhong, Yuxu论文数: 0 引用数: 0 h-index: 0机构: Beijing Inst Pharmacol & Toxicol, State Key Lab Toxicol & Med Countermeasures, Beijing 100850, Peoples R China Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R ChinaKong, Dexin论文数: 0 引用数: 0 h-index: 0机构: Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R China Tianjin Med Univ, Sch Pharmaceut Sci, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R China
- [2] Enhanced PI3K p110α Signaling Confers Acquired Lapatinib Resistance That Can Be Effectively Reversed by a p110α-Selective PI3K Inhibitor[J]. MOLECULAR CANCER THERAPEUTICS, 2014, 13 (01) : 60 - 70Brady, Samuel W.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USA Univ Texas Hlth Sci Ctr Houston, Grad Sch Biomed Sci, Canc Biol Program, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USAZhang, Jian论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USASeok, Daniel论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USAWang, Hai论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Dept Mol & Cellular Oncol, Houston, TX 77030 USA论文数: 引用数: h-index:机构:
- [3] Synthesis, biological evaluation and molecular modelling of sulfonohydrazides as selective PI3K p110α inhibitors[J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2007, 15 (24) : 7677 - 7687Kendall, Jackie D.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandRewcastle, Gordon W.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New Zealand Univ Auckland, Maurice Wilkins Ctr Mol Biodiscovery, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandFrederick, Raphael论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandMawson, Claire论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandDenny, William A.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New Zealand Univ Auckland, Maurice Wilkins Ctr Mol Biodiscovery, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandMarshall, Elaine S.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandBaguley, Bruce C.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandChaussade, Claire论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Dept Mol Med & Pathol, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandJackson, Shaun P.论文数: 0 引用数: 0 h-index: 0机构: Monash Univ, Australian Ctr Blood Dis, Melbourne, Vic 3004, Australia Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New ZealandShepherd, Peter R.论文数: 0 引用数: 0 h-index: 0机构: Univ Auckland, Sch Med & Hlth Sci, Dept Mol Med & Pathol, Auckland 1020, New Zealand Univ Auckland, Maurice Wilkins Ctr Mol Biodiscovery, Auckland 1020, New Zealand Univ Auckland, Sch Med & Hlth Sci, Auckland Canc Soc Res Ctr, Auckland 1020, New Zealand
- [4] Discovery of a Novel Series of Thienopyrimidine as Highly Potent and Selective PI3K Inhibitors[J]. ACS MEDICINAL CHEMISTRY LETTERS, 2015, 6 (04): : 434 - 438Han, Fangbin论文数: 0 引用数: 0 h-index: 0机构: PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R ChinaLin, Songwen论文数: 0 引用数: 0 h-index: 0机构: PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R ChinaLiu, Peng论文数: 0 引用数: 0 h-index: 0机构: PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R ChinaLiu, Xiujie论文数: 0 引用数: 0 h-index: 0机构: PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R ChinaTao, Jing论文数: 0 引用数: 0 h-index: 0机构: PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R ChinaDeng, Xiaobing论文数: 0 引用数: 0 h-index: 0机构: PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R ChinaYi, Chongqin论文数: 0 引用数: 0 h-index: 0机构: PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R ChinaXu, Heng论文数: 0 引用数: 0 h-index: 0机构: PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China PKUCare Pharmaceut R&D Ctr, Biotech Innovat Works, Beijing 102206, Peoples R China
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BLOOD, 2010, 116 (09) : 1460 - 1468Ikeda, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Sapporo Med Univ, Dept Internal Med 1, Sapporo, Hokkaido, Japan Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAHideshima, Teru论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAFulciniti, Mariateresa论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAPerrone, Giulia论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAMiura, Naoya论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAYasui, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Sapporo Med Univ, Dept Internal Med 1, Sapporo, Hokkaido, Japan Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAOkawa, Yutaka论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAKiziltepe, Tanyel论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USASanto, 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Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USARichardson, Paul论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAMunshi, Nikhil C.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Boston VA Healthcare Syst, W Roxbury, MA USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USALannutti, Brian J.论文数: 0 引用数: 0 h-index: 0机构: Calistoga Pharmaceut Inc, Seattle, WA USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAPuri, Kamal D.论文数: 0 引用数: 0 h-index: 0机构: Calistoga Pharmaceut Inc, Seattle, WA USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAGiese, Neill A.论文数: 0 引用数: 0 h-index: 0机构: Calistoga Pharmaceut Inc, Seattle, WA USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USAAnderson, Kenneth C.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA Harvard Univ, Sch Med, Lebow Inst Myeloma Therapeut, Boston, MA 02115 USA Harvard Univ, Sch Med, Dana Farber Canc Inst, Jerome Lipper Multiple Myeloma Ctr,Dept Med Oncol, Boston, MA 02115 USA
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