Discovery of novel and highly selective PI3Kδ inhibitors based on the p110δ crystal structure

被引:2
|
作者
Jia, Wen-Qing [1 ]
Liu, Ya-Ya [1 ]
Feng, Xiao-Yan [1 ]
Xu, Wei-Ren [2 ]
Cheng, Xian-Chao [1 ]
机构
[1] Tianjin Med Univ, Sch Pharm, Tianjin Key Lab Technol Enabling Dev Clin Therape, Tianjin 300070, Peoples R China
[2] Tianjin Inst Pharmaceut Res, Tianjin Key Lab Mol Design & Drug Discovery, Tianjin, Peoples R China
来源
基金
中国国家自然科学基金;
关键词
D O I
10.1080/07391102.2019.1635531
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:2499 / 2508
页数:10
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