Synthesis and in vitro anticancer activity of conjugates of MDP with Amino-acridine/acridone derivatives

被引：0
|
作者：
Gozdowska, M [1 ]
Dzierzbicka, K [1 ]
WysockaSkrzela, B [1 ]
Kolodziejczyk, AM [1 ]
机构：
[1] GDANSK TECH UNIV,DEPT DRUG TECHNOL & BIOCHEM,PL-80952 GDANSK,POLAND
来源：
POLISH JOURNAL OF CHEMISTRY | 1997年 / 71卷 / 06期
关键词：
amino-acridine/acridone derivatives; anticancer activity; muramyl dipeptide;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A series of MDP (muramyl dipeptide) analogues modified at the C-terminus of MDP molecule by the formation of an amide bond between the carboxylic group of isoglutamine and the amine function of the respective derivative of acridine or acridone were synthesized as potential anticancer agents.
引用
收藏
页码：767 / 773
页数：7
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