共 50 条
- [31] An inhibitor of ERK1/2 kinase acts as a potent modulator of conditioned aspects of drug-seeking behaviour in rats[J]. EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2011, 21 : S589 - S590Filip, M.论文数: 0 引用数: 0 h-index: 0机构: Jagiellonian Univ, Inst Pharmacol, Fac Pharm, Krakow, Poland Jagiellonian Univ, Inst Pharmacol, Fac Pharm, Krakow, PolandNowak, E.论文数: 0 引用数: 0 h-index: 0机构: Jagiellonian Univ, Inst Pharmacol, Fac Pharm, Krakow, Poland Jagiellonian Univ, Inst Pharmacol, Fac Pharm, Krakow, PolandPijanowska, A.论文数: 0 引用数: 0 h-index: 0机构: Jagiellonian Univ, Inst Pharmacol, Fac Pharm, Krakow, Poland Jagiellonian Univ, Inst Pharmacol, Fac Pharm, Krakow, PolandCzyzyk, J.论文数: 0 引用数: 0 h-index: 0机构: Jagiellonian Univ, Inst Pharmacol, Fac Pharm, Krakow, Poland Jagiellonian Univ, Inst Pharmacol, Fac Pharm, Krakow, Poland
- [32] Development of UCT-01-097, a novel orally available ERK1/2 inhibitor for the treatment of ERK1/2 dependent cancers[J]. CANCER RESEARCH, 2023, 83 (07)O'Brien, Neil A.论文数: 0 引用数: 0 h-index: 0McDermott, Martina S.论文数: 0 引用数: 0 h-index: 0O'Boyle, Brendan M.论文数: 0 引用数: 0 h-index: 0Reeves, Corey M.论文数: 0 引用数: 0 h-index: 0Bartberger, Michael论文数: 0 引用数: 0 h-index: 0Loson, Oliver论文数: 0 引用数: 0 h-index: 0Chau, Kevin论文数: 0 引用数: 0 h-index: 0Hong, Jenny J.论文数: 0 引用数: 0 h-index: 0Jia, Weiping论文数: 0 引用数: 0 h-index: 0Kamranpour, Naeimeh论文数: 0 引用数: 0 h-index: 0Luo, Tong论文数: 0 引用数: 0 h-index: 0Ayala, Raul论文数: 0 引用数: 0 h-index: 0Madrid, Athena M.论文数: 0 引用数: 0 h-index: 0Glaspy, John A.论文数: 0 引用数: 0 h-index: 0Stoltz, Brian M.论文数: 0 引用数: 0 h-index: 0Slamon, Dennis J.论文数: 0 引用数: 0 h-index: 0
- [33] Discovery of the Potent and Selective Inhaled Janus Kinase 1 Inhibitor AZD4604 and Its Preclinical Characterization[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2023, : 13400 - 13415Nilsson, Magnus论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenBerggren, Kristina论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenBerglund, Susanne论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenCerboni, Silvia论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenCollins, Mia论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenDahl, Goran论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Struct & Biophys Res & Early Dev, Discovery Sci, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenElmqvist, David论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Pharmaceut Sci, Early Prod Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenGrimster, Neil P.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Oncol R&D, Waltham, MA 02451 USA AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenHendrickx, Ramon论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Res & Early Dev, Resp & Immunol,DMPK, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenJohansson, Johan R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenKettle, Jason G.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Oncol R&D, Waltham, MA 02451 USA AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenLepisto, Matti论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenRhedin, Magdalena论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenSmailagic, Amir论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenSu, Qibin论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Oncol R&D, Waltham, MA 02451 USA AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenWennberg, Tiiu论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenWu, Allan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Discovery Sci, R&D, Waltham, MA 02451 USA AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenOsterlund, Torben论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Res & Early Dev, Discovery Sci,Mechanist Biol & Profiling, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenNaessens, Thomas论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, SwedenMitra, Suman论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Biosci Res & Early Dev, SE-43183 Gothenburg, Sweden AstraZeneca, BioPharmaceut R&D, Resp & Immunol, Med Chem Res & Early Dev, SE-43183 Gothenburg, Sweden
- [34] Discovery and Characterization of a Potent and Selective Inhibitor of Aedes aegypti Inward Rectifier Potassium Channels[J]. PLOS ONE, 2014, 9 (11):Raphemot, Rene论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USA Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USARouhier, Matthew F.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Ohio Agr Res & Dev Ctr, Dept Entomol, Wooster, OH 44691 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USASwale, Daniel R.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USADays, Emily论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Inst Chem Biol, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USAWeaver, C. David论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USALovell, Kimberly M.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Sch Med, Dept Chem, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USAKonkel, Leah C.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Sch Med, Dept Chem, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USAEngers, Darren W.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Sch Med, Dept Chem, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USABollinger, Sean F.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Sch Med, Dept Chem, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USAHopkins, Corey论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Sch Med, Dept Chem, Nashville, TN 37212 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USAPiermarini, Peter M.论文数: 0 引用数: 0 h-index: 0机构: Ohio State Univ, Ohio Agr Res & Dev Ctr, Dept Entomol, Wooster, OH 44691 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USADenton, Jerod S.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USA Vanderbilt Univ, Sch Med, Dept Pharmacol, Nashville, TN 37212 USA Vanderbilt Univ, Sch Med, Inst Chem Biol, Nashville, TN 37212 USA Vanderbilt Univ, Inst Global Hlth, Nashville, TN 37235 USA Vanderbilt Univ, Med Ctr, Dept Anesthesiol, Nashville, TN USA
- [35] Discovery and characterization of a potent and selective non-amidine inhibitor of human factor Xa[J]. BIOCHEMICAL PHARMACOLOGY, 2003, 65 (09) : 1407 - 1418Liang, AA论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USALight, DR论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USAKochanny, M论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USARumennik, G论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USATrinh, L论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USALentz, D论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USAPost, J论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USAMorser, J论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USASnider, M论文数: 0 引用数: 0 h-index: 0机构: Berlex Biosci, Richmond, CA 94806 USA Berlex Biosci, Richmond, CA 94806 USA
- [36] Discovery and characterization of the potent, selective and orally bioavailable MMP inhibitor ABT-770[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2001, 11 (12) : 1557 - 1560Curtin, ML论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAFlorjancic, AS论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAHeyman, HR论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAMichaelides, MR论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAGarland, RB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAHolms, JH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USASteinman, DH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USADellaria, JF论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAGong, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAWada, CK论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAGuo, Y论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAElmore, IB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USATapang, P论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAAlbert, DH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAMagoc, TJ论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAMarcotte, PA论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USABouska, JJ论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAGoodfellow, CL论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USABauch, JL论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAMarsch, KC论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USAMorgan, DW论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USADavidsen, SK论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA Abbott Labs, Canc Res Area, Dept 47J, Abbott Pk, IL 60064 USA
- [37] Discovery of a Potent and Selective DDR1 Receptor Tyrosine Kinase Inhibitor[J]. ACS CHEMICAL BIOLOGY, 2013, 8 (10) : 2145 - 2150Kim, Hyung-Gu论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USA Harvard Univ, Sch Med, Charlestown, MA 02129 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USATan, Li论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USAWeisberg, Ellen L.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USALiu, Feiyang论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Chinese Acad Sci, High Field Magnet Lab, Hefei 230031, Anhui, Peoples R China Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USA论文数: 引用数: h-index:机构:Choi, Hwan Geun论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USAEzell, Scott A.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USA Harvard Univ, Sch Med, Charlestown, MA 02129 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USAWu, Hong论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Chinese Acad Sci, High Field Magnet Lab, Hefei 230031, Anhui, Peoples R China Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USAZhao, Zheng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, High Field Magnet Lab, Hefei 230031, Anhui, Peoples R China Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USAWang, Jinhua论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USAMandinova, Anna论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USA Harvard Univ, Sch Med, Charlestown, MA 02129 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USAGriffin, James D.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USABullock, Alex N.论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Struct Genom Consortium, Oxford OX3 7DQ, England Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USALiu, Qingsong论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Chinese Acad Sci, High Field Magnet Lab, Hefei 230031, Anhui, Peoples R China Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USALee, Sam W.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USA Harvard Univ, Sch Med, Charlestown, MA 02129 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Harvard Univ, Sch Med, Dana Farber Canc Inst, Boston, MA 02115 USA Harvard Univ, Sch Med, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Massachusetts Gen Hosp, Cutaneous Biol Res Ctr, Charlestown, MA 02129 USA
- [38] Discovery of S64315, a Potent and Selective Mcl-1 Inhibitor[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (22) : 13762 - 13795Szlavik, Zoltan论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryCsekei, Marton论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryPaczal, Attila论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungarySzabo, Zoltan B.论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungarySipos, Szabolcs论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryRadics, Gabor论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryProszenyak, Agnes论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryBalint, Balazs论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, HungaryMurray, James论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryDavidson, James论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryChen, Ijen论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryDokurno, Pawel论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungarySurgenor, Allan E.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryDaniels, Zoe Marie论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryHubbard, Roderick E.论文数: 0 引用数: 0 h-index: 0机构: Vernalis R&D Ltd, Cambridge CB21 6GB, England Servier Res Inst Med Chem, H-1031 Budapest, HungaryLe Toumelin-Braizat, Gaetane论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryClaperon, Audrey论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryLysiak-Auvity, Gaelle论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryGirard, Anne-Marie论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryBruno, Alain论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryChanrion, Maia论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryColland, Frederic论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryMaragno, Ana-Leticia论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryDemarles, Didier论文数: 0 引用数: 0 h-index: 0机构: Technol Servier, F-45000 Orleans, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryGeneste, Olivier论文数: 0 引用数: 0 h-index: 0机构: Inst Rech Servier, F-78290 Croissy Sur Seine, France Servier Res Inst Med Chem, H-1031 Budapest, HungaryKotschy, Andras论文数: 0 引用数: 0 h-index: 0机构: Servier Res Inst Med Chem, H-1031 Budapest, Hungary Servier Res Inst Med Chem, H-1031 Budapest, Hungary
- [39] Discovery of a Potent, Selective, and Cell-Active SPIN1 Inhibitor[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2024, 67 (07) : 5837 - 5853Xiong, Yan论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Neurosci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAGreschik, Holger论文数: 0 引用数: 0 h-index: 0机构: Univ Freiburg, Dept Urol, Med Ctr, D-79106 Freiburg, Germany Univ Freiburg, Ctr Clin Res, Med Ctr, D-79106 Freiburg, Germany Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAJohansson, Catrine论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Botnar Res Ctr, Struct Genom Consortium, NIHR Oxford BRU, Oxford OX3 7LD, England Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USASeifert, Ludwig论文数: 0 引用数: 0 h-index: 0机构: Univ Freiburg, Inst Pharmaceut Sci, D-79104 Freiburg, Germany Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAGamble, Vicki论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Botnar Res Ctr, Struct Genom Consortium, NIHR Oxford BRU, Oxford OX3 7LD, England Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAPark, Kwang-su论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Neurosci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAFagan, Vincent论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Ctr Med Discovery, Nuffield Dept Med, Oxford OX3 7FZ, England Univ Oxford, Target Discovery Inst, Nuffield Dept Med, Oxford OX3 7FZ, England Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USA论文数: 引用数: h-index:机构:Chau, Irene论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAVedadi, Masoud论文数: 0 引用数: 0 h-index: 0机构: Ontario Inst Canc Res, Toronto, ON M5G 0A3, Canada Univ Toronto, Dept Pharmacol & Toxicol, Toronto, ON M5S 1A8, Canada Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAArrowsmith, Cheryl H.论文数: 0 引用数: 0 h-index: 0机构: Univ Toronto, Struct Genom Consortium, Toronto, ON M5G 1L7, Canada Univ Toronto, Princess Margaret Canc Ctr, Toronto, ON M5G 1L7, Canada Univ Toronto, Dept Med Biophys, Toronto, ON M5G 1L7, Canada Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USABrennan, Paul论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Ctr Med Discovery, Nuffield Dept Med, Oxford OX3 7FZ, England Univ Oxford, Target Discovery Inst, Nuffield Dept Med, Oxford OX3 7FZ, England Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAFedorov, Oleg论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Ctr Med Discovery, Nuffield Dept Med, Oxford OX3 7FZ, England Univ Oxford, Target Discovery Inst, Nuffield Dept Med, Oxford OX3 7FZ, England Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAJung, Manfred论文数: 0 引用数: 0 h-index: 0机构: Univ Freiburg, Inst Pharmaceut Sci, D-79104 Freiburg, Germany German Canc Res Ctr, D-69120 Heidelberg, Germany German Canc Consortium DKTK, Freiburg, Germany Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAFarnie, Gillian论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Ctr Med Discovery, Nuffield Dept Med, Oxford OX3 7FZ, England Univ Oxford, Target Discovery Inst, Nuffield Dept Med, Oxford OX3 7FZ, England Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USALiu, Jing论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Oncol Sci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Neurosci, New York, NY 10029 USA Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAOppermann, Udo论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Botnar Res Ctr, Struct Genom Consortium, NIHR Oxford BRU, Oxford OX3 7LD, England Univ Oxford, Botnar Res Ctr, Oxford OX3 7LD, England Univ Oxford, Oxford Ctr Translat Myeloma Res, Oxford OX3 7LD, England Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USASchuele, Roland论文数: 0 引用数: 0 h-index: 0机构: Univ Freiburg, Dept Urol, Med Ctr, D-79106 Freiburg, Germany Univ Freiburg, Ctr Clin Res, Med Ctr, D-79106 Freiburg, Germany German Canc Consortium DKTK, Freiburg, Germany Univ Freiburg, CIBSS Ctr Biol Signalling Studies, Freiburg, Germany Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USAJin, Jian论文数: 0 引用数: 0 h-index: 0机构: Icahn Sch Med Mt Sinai, Tisch Canc Inst, Mt Sinai Ctr Therapeut Discovery, Dept Pharmacol Sci, New York, NY 10029 USA Icahn Sch Med 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- [40] Discovery of the first potent and selective Mycobacterium tuberculosis Zmp1 inhibitor[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (11) : 2508 - 2511论文数: 引用数: h-index:机构:Moraca, Francesca论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, ItalyDeodato, Davide论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, ItalyFerraris, Davide M.论文数: 0 引用数: 0 h-index: 0机构: Univ Piemonte Orientale, Dipartimento Sci Farmaco, I-28100 Novara, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, ItalySelchow, Petra论文数: 0 引用数: 0 h-index: 0机构: Univ Zurich, Inst Med Microbiol, CH-8006 Zurich, Switzerland Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, ItalySander, Peter论文数: 0 引用数: 0 h-index: 0机构: Univ Zurich, Inst Med Microbiol, CH-8006 Zurich, Switzerland NRLM, CH-8006 Zurich, Switzerland Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, ItalyRizzi, Menico论文数: 0 引用数: 0 h-index: 0机构: Univ Piemonte Orientale, Dipartimento Sci Farmaco, I-28100 Novara, Italy Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, ItalyBotta, Maurizio论文数: 0 引用数: 0 h-index: 0机构: Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, Italy Temple Univ, Coll Sci & Technol, Sbarro Inst Canc Res & Mol Med, Ctr Biotechnol, Philadelphia, PA 19122 USA Univ Siena, Dipartimento Biotecnol Chim & Farm, I-53100 Siena, Italy