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- [1] Discovery of GDC-0994, a potent and selective ERK1/2 inhibitor in early clinical development[J]. CANCER RESEARCH, 2014, 74 (19)Robarge, Kirk论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USASchwarz, Jacob论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USABlake, Jim论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USABurkard, Michael论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAChan, Jocelyn论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAChen, Huifen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAChou, Kang-Jye论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USADiaz, Dolores论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAGaudino, John论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAGould, Stephen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAGrina, Jonas论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAXin Linghu论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USALiu, Lichuan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAMartinson, Matthew论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAMoreno, David A.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAOrr, Christine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAPacheco, Patricia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAQin, Ann论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USARasor, Kevin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USARen, Li论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAShahidi-Latham, Sheerin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAStults, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USASullivan, Francis论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAWang, Weiru论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAYin, Peter论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAZhou, Aihe论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USABelvin, Marcia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAMerchant, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAMoffat, John G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Array Biopharma, Boulder, CO USA Genentech Inc, San Francisco, CA USA
- [2] Discovery of GDC-0994, a potent and selective ERK1/2 inhibitor in early clinical development[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 252Schwarz, Jacob论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USABlake, James论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USABurkard, Michael论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAChan, Jocelyn论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAChen, Huifen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAChou, Kang-Jye论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USADiaz, Dolores论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USADudley, Danette论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAGaudino, John论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAGould, Stephen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAGrina, Jonas论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAHunsaker, Thomas论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USALiu, Lichuan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAMartinson, Matthew论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAMoreno, David论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAOrr, Christine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAPacheco, Patricia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAQin, Ann论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USARasor, Kevin论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USARen, Li论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USARobarge, Kirk论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAShahidi-Latham, Sheerin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAStults, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USASullivan, Francis论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO USA Genentech Inc, San Francisco, CA USAWang, Weiru论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAYin, Jianping论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAZhou, Aihe论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USABelvin, Marcia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAMerchant, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAMoffat, John论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USA
- [3] Discovery of potent and selective inhibitors of ERK1/2 with a unique mechanism of action[J]. CANCER RESEARCH, 2016, 76Deng, Yongqi论文数: 0 引用数: 0 h-index: 0Samatar, Ahmed论文数: 0 引用数: 0 h-index: 0Shipps, Gerald论文数: 0 引用数: 0 h-index: 0Cooper, Alan论文数: 0 引用数: 0 h-index: 0Long, Brian论文数: 0 引用数: 0 h-index: 0Carr, Donnar论文数: 0 引用数: 0 h-index: 0Xiao, Li论文数: 0 引用数: 0 h-index: 0Hruza, Alan论文数: 0 引用数: 0 h-index: 0Wang, Tong论文数: 0 引用数: 0 h-index: 0Zhu, Liang论文数: 0 引用数: 0 h-index: 0Nan, Yang论文数: 0 引用数: 0 h-index: 0Patel, Mehul论文数: 0 引用数: 0 h-index: 0Muppalla, Kiran论文数: 0 引用数: 0 h-index: 0Zhu, Hugh论文数: 0 引用数: 0 h-index: 0Boga, Babu Sobhana论文数: 0 引用数: 0 h-index: 0Gao, Xiaolei论文数: 0 引用数: 0 h-index: 0
- [4] Discovery of Highly Potent, Selective, and Efficacious Small Molecule Inhibitors of ERK1/2[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2015, 58 (04) : 1976 - 1991Ren, Li论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAGrina, Jonas论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAMoreno, David论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USABlake, James F.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAGaudino, John J.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAGarrey, Rustam论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAMetcalf, Andrew T.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USABurkard, Michael论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAMartinson, Matthew论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USARasor, Kevin论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Array BioPharma Inc, Boulder, CO 80301 USAChen, Huifen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USADean, Brian论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAGould, Stephen E.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAPacheco, Patricia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAShahidi-Latham, Sheerin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAYin, Jianping论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAWest, Kristina论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAWang, Weiru论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USAMoffat, John G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USASchwarz, Jacob B.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Array BioPharma Inc, Boulder, CO 80301 USA
- [5] Discovery and characterization of AZ285 as a potent and selective inhibitor of CK2 kinase[J]. CANCER RESEARCH, 2012, 72Dowling, James E.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USAAlimzhanov, Marat论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USABao, Larry论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USABrassil, Patrick论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USACooke, Emma L.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USADenz, Christopher R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USALiu, Zhong-Ying论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USAYe, Qing论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USALyne, Paul D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Waltham, MA USA AstraZeneca, Waltham, MA USA
- [6] Fragment-based discovery of a highly potent, orally bioavailable ERK1/2 inhibitor that modulates the phosphorylation and catalytic activity of ERK1/2[J]. MOLECULAR CANCER THERAPEUTICS, 2018, 17 (01)Heightman, Tom D.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandBerdini, Valerio论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandBraithwaite, Hannah论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandBuck, Ildiko论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandCassidy, Megan论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandCastro, Juan论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandCourtin, Aurelie论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandDay, James论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandEast, Charlotte论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandFazal, Lynsey论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandGraham, Brent论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandGriffiths-Jones, Charlotte论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandLyons, John论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandMartins, Vanessa论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandMuench, Sandra论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandMunck, Joanne论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandNorton, David论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandO'Reilly, Marc论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandPalmer, Nick论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandPathuri, Puja论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandReader, Mike论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandRees, David论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandRich, Sharna论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandRichardson, Caroline论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandSaini, Harpreet论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandThompson, Neil论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandWallis, Nicola论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandWalton, Hugh论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandWilsher, Nicola论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandWoolford, Alison论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, EnglandMurray, Chris论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut Inc, Cambridge, England Astex Pharmaceut Inc, Cambridge, England
- [7] Preclinical characterization of HMPL-295, a potent and selective ERK 1/2 inhibitor[J]. CANCER RESEARCH, 2024, 84 (06)Hu, Jia论文数: 0 引用数: 0 h-index: 0Ni, Jun论文数: 0 引用数: 0 h-index: 0Lv, Yuanzhi论文数: 0 引用数: 0 h-index: 0Li, Wenjun论文数: 0 引用数: 0 h-index: 0Zhang, Hui论文数: 0 引用数: 0 h-index: 0Li, Xin论文数: 0 引用数: 0 h-index: 0Yu, Ying论文数: 0 引用数: 0 h-index: 0Zhong, Zeyu论文数: 0 引用数: 0 h-index: 0Wang, Jian论文数: 0 引用数: 0 h-index: 0Sai, Yang论文数: 0 引用数: 0 h-index: 0Qing, Weiguo论文数: 0 引用数: 0 h-index: 0Ren, Yongxin论文数: 0 引用数: 0 h-index: 0Shi, Michael论文数: 0 引用数: 0 h-index: 0Su, Weiguo论文数: 0 引用数: 0 h-index: 0
- [8] Discovery of AZD0364, a potent and selective oral inhibitor of ERK1/2 that is efficacious in both monotherapy and combination therapy in models of NSCLC[J]. CANCER RESEARCH, 2018, 78 (13)Simpson, Iain论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandAnderton, Mark J.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandAndrews, David M.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandBreed, Jason论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandDavies, Emma论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandDebreczeni, Judit E.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandFlemington, Vikki论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandGibbons, Francis D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Boston, MA USA AstraZeneca, Cambridge, EnglandGraham, Mark A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandHopcroft, Philip论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandHoward, Tina论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandHudson, Julian论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandJones, Clifford D.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandJones, Christopher论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandLindsay, Nicola论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandPease, J. Elizabeth论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandRawlins, Philip论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandRoberts, Karen论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandSwallow, Steve论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandSt-Gallay, Steve论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandTonge, Michael E.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, EnglandWard, Richard A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Cambridge, England AstraZeneca, Cambridge, England
- [9] Discovery of LY3214996, a selective and novel ERK1/2 inhibitor with potent antitumor activities in cancer models with MAPK pathway alterations[J]. CANCER RESEARCH, 2017, 77Bhagwat, Shripad V.论文数: 0 引用数: 0 h-index: 0McMillen, William T.论文数: 0 引用数: 0 h-index: 0Cai, Shufen论文数: 0 引用数: 0 h-index: 0Zhao, Baohui论文数: 0 引用数: 0 h-index: 0Whitesell, Matthew论文数: 0 引用数: 0 h-index: 0Kindler, Lisa论文数: 0 引用数: 0 h-index: 0Flack, Robert S.论文数: 0 引用数: 0 h-index: 0Wu, Wenjuan论文数: 0 引用数: 0 h-index: 0Huss, Karen论文数: 0 引用数: 0 h-index: 0Anderson, Bryan论文数: 0 引用数: 0 h-index: 0Yuan, Xiu-Juan论文数: 0 引用数: 0 h-index: 0Jaken, Susan论文数: 0 引用数: 0 h-index: 0McCann, Denis论文数: 0 引用数: 0 h-index: 0Mathes, Brian论文数: 0 引用数: 0 h-index: 0Dropsey, Andrew J.论文数: 0 引用数: 0 h-index: 0Manro, Jason论文数: 0 引用数: 0 h-index: 0Walgren, Jennie论文数: 0 引用数: 0 h-index: 0Yuen, Eunice论文数: 0 引用数: 0 h-index: 0Gong, Xueqian论文数: 0 引用数: 0 h-index: 0Rodriguez, Michael J.论文数: 0 引用数: 0 h-index: 0Huang, Jianping论文数: 0 引用数: 0 h-index: 0Tiu, Ramon V.论文数: 0 引用数: 0 h-index: 0Joseph, Sajan论文数: 0 引用数: 0 h-index: 0Peng, Sheng-Bin论文数: 0 引用数: 0 h-index: 0
- [10] Characterization of a novel ERK1/2 inhibitor, which modulates the phosphorylation and catalytic activity of ERK1/2[J]. MOLECULAR CANCER THERAPEUTICS, 2018, 17 (01)Munck, Joanne M.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandBerdini, Valerio论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandBevan, Luke D.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandBraithwaite, Hannah论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandBuck, Ildiko M.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandCassidy, Megan论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandCastro, Juan论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandCourtin, Aurelie论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandDay, James E.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandEast, Charlotte论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandFazal, Lynsey论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandGraham, Brent论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandGriffiths-Jones, Charlotte M.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandHeightman, Tom D.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandHindley, Chris J.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandKidane, Birikiti论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandKucia-Tran, Justyna论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandLyons, John F.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandMartins, Vanessa论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandMuench, Sandra论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandMurray, Chris W.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandNorton, David论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandO'Reilly, Marc论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandPalmer, Nick论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandPathuri, Puja论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandReader, Mike论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandRees, David C.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandRich, Sharna J.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandRichardson, Caroline J.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandSaini, Harpreet K.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandShah, Alpesh论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandStanczuk, Lukas论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandThompson, Neil T.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandWalton, Hugh论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandWilsher, Nicola E.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandWoolford, Alison J.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, EnglandWallis, Nicola G.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge, England Astex Pharmaceut, Cambridge, England