A transgenic mouse model for in vivo regulation of the human CYP3A4 promoter

被引:0
|
作者
Zhang, WS [1 ]
Purchio, A [1 ]
Chen, K [1 ]
Wu, JM [1 ]
Lu, L [1 ]
West, DB [1 ]
机构
[1] Xenogen Corp, Alameda, CA 94501 USA
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
235
引用
收藏
页码:118 / 118
页数:1
相关论文
共 50 条
  • [31] Contribution of metabolites to in vivo CYP3A4 inhibition by itraconazole
    Templeton, Ian E.
    Thummel, Kenneth E.
    Isoherranen, Nina
    Kharasch, Evan David
    Kunze, Kent L.
    Nelson, Wendel L.
    Hoffer, Christine
    DRUG METABOLISM REVIEWS, 2006, 38 : 127 - 128
  • [32] Effect of a CYP3A4 promoter variant on a reporter gene.
    Amirimani, B
    Walker, AH
    Weber, BL
    Rebbeck, TR
    AMERICAN JOURNAL OF HUMAN GENETICS, 1999, 65 (04) : A181 - A181
  • [33] Regulation of CYP3A4 by the bile acid receptor FXR:: evidence for functional binding sites in the CYP3A4 gene
    Gnerre, C
    Blättler, S
    Kaufmann, MR
    Looser, R
    Meyer, UA
    PHARMACOGENETICS, 2004, 14 (10): : 635 - 645
  • [34] Contribution of itraconazole metabolites to inhibition of CYP3A4 in vivo
    Templeton, I. E.
    Thummel, K. E.
    Kharasch, E. D.
    Kunze, K. L.
    Hoffer, C.
    Nelson, Wl
    Isoherranen, N.
    CLINICAL PHARMACOLOGY & THERAPEUTICS, 2008, 83 (01) : 77 - 85
  • [35] Effect of influenza immunization on CYP3A4 activity in vivo
    Hayney, MS
    Muller, D
    JOURNAL OF CLINICAL PHARMACOLOGY, 2003, 43 (12): : 1377 - 1381
  • [36] Bufalin inhibits CYP3A4 activity in vitro and in vivo
    Hai-yun Li
    Wen Xu
    Xi Zhang
    Wei-dong Zhang
    Li-wei Hu
    Acta Pharmacologica Sinica, 2009, 30 : 646 - 652
  • [37] DNA methylation dynamics in the hepatic CYP3A4 gene promoter
    Kacevska, Marina
    Ivanov, Maxim
    Wyss, Annika
    Kasela, Silva
    Milani, Lili
    Rane, Anders
    Ingelman-Sundberg, Magnus
    BIOCHIMIE, 2012, 94 (11) : 2338 - 2344
  • [38] Transcriptional regulation of CYP3A4 by nuclear receptors in human hepatocytes under hypoxia
    Yuan, Xuechun
    Lu, Hui
    Zhao, Anpeng
    Ding, Yidan
    Min, Qiong
    Wang, Rong
    DRUG METABOLISM REVIEWS, 2020, 52 (02) : 225 - 234
  • [39] In Vitro-In Vivo Inaccuracy: The CYP3A4 Anomaly
    Bowman, Christine M.
    Benet, Leslie Z.
    DRUG METABOLISM AND DISPOSITION, 2019, 47 (12) : 1368 - 1371
  • [40] Bufalin inhibits CYP3A4 activity in vitro and in vivo
    Li, Hai-yun
    Xu, Wen
    Zhang, Xi
    Zhang, Wei-dong
    Hu, Li-wei
    ACTA PHARMACOLOGICA SINICA, 2009, 30 (05) : 646 - 652