Computational design of a high-activity mutant of human butyrylcholinesterase specific for treatment of cocaine abuse

被引:0
|
作者
Zheng, Fang [1 ]
Xue, Liu [1 ]
Hou, Shurong [1 ]
Yang, Wenchao [1 ]
Zhan, Max [1 ]
Zhan, Chang-Guo [1 ]
机构
[1] Univ Kentucky, Dept Pharmaceut Sci, Lexington, KY 40536 USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
236-COMP
引用
收藏
页数:1
相关论文
共 50 条
  • [21] Design and expression of organophosphorus acid anhydride hydrolase activity in human butyrylcholinesterase
    Millard, CB
    Lockridge, O
    Broomfield, CA
    BIOCHEMISTRY, 1995, 34 (49) : 15925 - 15933
  • [22] High activity of human butyrylcholinesterase at low pH in the presence of excess butyrylthiocholine
    Masson, P
    Nachon, F
    Bartels, CF
    Froment, MT
    Ribes, F
    Matthews, C
    Lockridge, O
    EUROPEAN JOURNAL OF BIOCHEMISTRY, 2003, 270 (02): : 315 - 324
  • [23] A synthesis of [3H] cocaine at high specific activity
    Filer, Crist N.
    JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY, 2024, 333 (10) : 4869 - 4872
  • [24] Mechanical aspects of the phosphotriesterase activity of human butyrylcholinesterase G11 7H mutant
    Albaret, C
    Masson, P
    Broomfield, CA
    El Kaim, L
    Fortier, PL
    STRUCTURE AND FUNCTION OF CHOLINESTERASES AND RELATED PROTEINS, 1998, : 399 - 405
  • [25] ISOLATION AND PROPERTIES OF A HIGH-ACTIVITY LUCIFERASE FROM AN ALDEHYDE-REQUIRING MUTANT OF VIBRIO-HARVEYI
    AHMAD, M
    LEE, J
    FEDERATION PROCEEDINGS, 1985, 44 (04) : 1216 - 1216
  • [26] TREATMENT OF MALIGNANT BRAIN-TUMORS WITH HIGH-ACTIVITY I125
    WARA, WM
    GUTIN, PA
    LEIBEL, SA
    WEAVER, KA
    LAMB, S
    JOURNAL OF NEURO-ONCOLOGY, 1984, 2 (03) : 284 - 284
  • [27] PRODUCTION OF HIGH-ACTIVITY TC-99M GENERATORS FOR HUMAN USE
    MILENKOVIC, SM
    VUCINA, JL
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE, 1984, 9 (07): : A57 - A57
  • [28] Au-Decorated Silicene: Design of a High-Activity Catalyst toward CO Oxidation
    Li, Chong
    Yang, Shengxue
    Li, Shu-Shen
    Xia, Jian-Bai
    Li, Jingbo
    JOURNAL OF PHYSICAL CHEMISTRY C, 2013, 117 (01): : 483 - 488
  • [29] A fluorescent probe for butyrylcholinesterase activity in human serum based on a fluorophore with specific binding affinity for human serum albumin
    Yoo, Soyeon
    Han, Min Su
    CHEMICAL COMMUNICATIONS, 2019, 55 (97) : 14574 - 14577
  • [30] A Grafting Strategy for the Design of Improved G-Quadruplex Aptamers and High-Activity DNAzymes
    Li, Tao
    Wang, Erkang
    Dong, Shaojun
    PLOS ONE, 2009, 4 (04):