Reaction of 2-(nitroamino)pyrimidin-4(3H)-one derivatives with arylamines of low basicity in pivalic acid

被引：2
|
作者：
Novakov, I. A. [1 ]
Babushkin, A. S. [1 ]
Brunilina, L. L. [1 ]
Navrotskii, M. B. [1 ]
Orlinson, B. S. [1 ]
Robinovich, M. D. [1 ]
Yablokov, A. S. [1 ]
机构：
[1] Volgograd State Tech Univ, Pr Lenina 28, Volgograd 400005, Russia
来源：
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2016年 / 52卷 / 11期
基金：
俄罗斯基础研究基金会;
关键词：
AGENTS;
D O I：
10.1134/S1070428016110178
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Pivalic acid was used as a solvent for aminolysis of poly-substituted 2-(nitroamino)-pyrimidin-4(3De)-one derivatives with arylamines of low basicity. The reaction did not occur in the other solvents or without solvent. Aminolysis products were obtained in 51-59% yields.
引用
收藏
页码：1654 / 1656
页数：3
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