Prediction of human pharmacokinetics based on preclinical in vitro and in vivo data

被引:0
|
作者
Lavé, T [1 ]
Luttringer, O [1 ]
Zuegge, J [1 ]
Schneider, G [1 ]
Coassolo, R [1 ]
Theil, FR [1 ]
机构
[1] F Hoffmann La Roche Inc, Drug Discovery Support, CH-4070 Basel, Switzerland
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:81 / 104
页数:24
相关论文
共 50 条
  • [1] Practical Anticipation of Human Efficacious Doses and Pharmacokinetics Using In Vitro and Preclinical In Vivo Data
    Heimbach, Tycho
    Lakshminarayana, Suresh B.
    Hu, Wenyu
    He, Handan
    AAPS JOURNAL, 2009, 11 (03): : 602 - 614
  • [2] Practical Anticipation of Human Efficacious Doses and Pharmacokinetics Using In Vitro and Preclinical In Vivo Data
    Tycho Heimbach
    Suresh B. Lakshminarayana
    Wenyu Hu
    Handan He
    The AAPS Journal, 2009, 11 : 602 - 614
  • [3] Application of In Silico, In Vitro and Preclinical Pharmacokinetic Data for the Effective and Efficient Prediction of Human Pharmacokinetics
    Grime, Kenneth H.
    Barton, Patrick
    McGinnity, Dermot F.
    MOLECULAR PHARMACEUTICS, 2013, 10 (04) : 1191 - 1206
  • [4] Prediction of in vivo drug disposition from in vitro data based on physiological pharmacokinetics
    Iwatsubo, T
    Hirota, N
    Ooie, T
    Suzuki, H
    Sugiyama, Y
    BIOPHARMACEUTICS & DRUG DISPOSITION, 1996, 17 (04) : 273 - 310
  • [5] Recent developments in in vitro and in vivo models for improved translation of preclinical pharmacokinetics and pharmacodynamics data
    Yadav, Jaydeep
    El Hassani, Mehdi
    Sodhi, Jasleen
    Lauschke, Volker M.
    Hartman, Jessica H.
    Russell, Laura E.
    DRUG METABOLISM REVIEWS, 2021, 53 (02) : 207 - 233
  • [6] PREDICTION OF HUMAN PHARMACOKINETICS OF EPITINIB FROM PRECLINICAL PHARMACOKINETICS BY A PHYSIOLOGICALLY BASED PHARMACOKINETIC MODEL
    Ren, Hongcan
    Gu, Yi
    Wang, Jian
    Ni, Liang
    Zhang, Weijun
    Zhang, Li
    Tang, Xianli
    Gu, Dongxia
    Zhao, Jingjing
    Xu, Xiaoyan
    Yang, Haibin
    Zhang, Weihan
    Su, Weiguo
    Sai, Yang
    DRUG METABOLISM REVIEWS, 2014, 45 : 110 - 111
  • [7] The prediction of human pharmacokinetic parameters from preclinical and in vitro metabolism data
    Obach, RS
    Baxter, JG
    Liston, TE
    Silber, BM
    Jones, BC
    MacIntyre, F
    Rance, DJ
    Wastall, P
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 1997, 283 (01): : 46 - 58
  • [8] PRECLINICAL PHARMACOKINETICS OF NATURAL ANTIBIOTIC NEGAMYCIN AND PREDICTION OF ITS PHARMACOKINETICS IN HUMAN
    Guo, Jian
    Miele, Eric
    Luzietti, Ricardo A.
    Walsky, Robert L.
    DRUG METABOLISM REVIEWS, 2015, 47 : 218 - 218
  • [9] Predicting human pharmacokinetics from preclinical data
    Poggesi, I
    CURRENT OPINION IN DRUG DISCOVERY & DEVELOPMENT, 2004, 7 (01) : 100 - 111
  • [10] Benchmarking of Human Dose Prediction for Inhaled Medicines from Preclinical In Vivo Data
    Ericsson, Therese
    Friden, Markus
    Karrman-Mardh, Carina
    Dainty, Ian
    Grime, Ken
    PHARMACEUTICAL RESEARCH, 2017, 34 (12) : 2557 - 2567