Down-regulation of A2A coronary adenosine receptors by ZM-241385 and SCH-58261.

被引:0
|
作者
Rekik, M [1 ]
Mustafa, SJ [1 ]
机构
[1] E Carolina Univ, Sch Med, Dept Pharmacol, Greenville, NC 27858 USA
来源
FASEB JOURNAL | 2000年 / 14卷 / 04期
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:A165 / A165
页数:1
相关论文
共 50 条
  • [21] [3H]-ZM 241385 binding to endogenous A2A adenosine receptors is regulated by agonist pretreatment and GRK2
    Willets, JM
    Matharu, AL
    Kelly, E
    BRITISH JOURNAL OF PHARMACOLOGY, 2000, 129 : U136 - U136
  • [22] Structure of the Adenosine A2A Receptor in Complex with ZM241385 and the Xanthines XAC and Caffeine
    Dore, Andrew S.
    Robertson, Nathan
    Errey, James C.
    Ng, Irene
    Hollenstein, Kaspar
    Tehan, Ben
    Hurrell, Edward
    Bennett, Kirstie
    Congreve, Miles
    Magnani, Francesca
    Tate, Christopher G.
    Weir, Malcolm
    Marshall, Fiona H.
    STRUCTURE, 2011, 19 (09) : 1283 - 1293
  • [23] Kinetic and functional properties of [3H]ZM241385, a high affinity antagonist for adenosine A2A receptors
    Uustare, A
    Vonk, A
    Terasmaa, A
    Fuxe, K
    Rinken, A
    LIFE SCIENCES, 2005, 76 (13) : 1513 - 1526
  • [24] Binding of the antagonist radioligand [3H]-ZM241385 to A2A adenosine receptors in rat brain homogenates
    Alexander, SPH
    BRITISH JOURNAL OF PHARMACOLOGY, 1998, 125 : U15 - U15
  • [25] Iron deficiency in rats results in functional up-regulation of adenosine A2A receptors and functional down-regulation of adenosine A1 receptors
    Pearson, V
    Quiroz, C.
    Gulyani, S.
    Allen, R. P.
    Earley, C. J.
    Ferre, S.
    SLEEP, 2008, 31 : A266 - A266
  • [26] ZM 241385, an adenosine A2A receptor antagonist, inhibits hippocampal A1 receptor responses
    Lopes, LV
    Cunha, RA
    Ribeiro, JA
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1999, 383 (03) : 395 - 398
  • [27] Biaryl and heteroaryl derivatives of SCH 58261 as potent and selective adenosine A2A receptor antagonists
    Shah, Unmesh
    Boyle, Craig D.
    Chackalamannil, Samuel
    Neustadt, Bernard R.
    Lindo, Neil
    Greenlee, William J.
    Foster, Carolyn
    Arik, Leyla
    Zhai, Ying
    Ng, Kwokei
    Wang, Shiyong
    Monopoli, Angela
    Lachowicz, Jean E.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (14) : 4199 - 4203
  • [28] Characterization of [125I]ZM241385 binding to adenosine A2A receptors in pineal gland of sheep brain.
    Koos, BJ
    Yan, XZ
    Kruger, L
    Linden, J
    Murray, TF
    JOURNAL OF THE SOCIETY FOR GYNECOLOGIC INVESTIGATION, 2006, 13 (02) : 304A - 304A
  • [29] Autoradiographic analysis of the binding of the antagonist radioligand [3H]-ZM241385 to A2A adenosine receptors in rat striatum
    Millns, P
    Alexander, SPH
    BRITISH JOURNAL OF PHARMACOLOGY, 1999, 128 : U81 - U81
  • [30] Biaryl and heteroaryl derivatives of SCH 58261 as potent and selective adenosine A2A receptor antagonists
    Shah, U
    Boyle, CD
    Chackalamannil, S
    Neustadt, B
    Foster, C
    Arik, L
    Zhai, Y
    Lachowicz, JE
    Ng, K
    Shiyong, W
    Monopoli, A
    Ongini, E
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U2549 - U2550