Synthesis of substituted 5,6-dihydro-4H[1,2,4]triazolo[4,3-a][1,5]benzodiazepines

被引:0
|
作者
Kosychova, L [1 ]
Stumbreviciute, Z [1 ]
Pleckaitiene, L [1 ]
Janciene, R [1 ]
Poudziunaite, BD [1 ]
机构
[1] Inst Biochem, LT-2600 Vilnius, Lithuania
关键词
4-acylhydrazino-2,3-dihydro-1H-1,5-benzodiazepines; 4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepines; cyclization;
D O I
暂无
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
An one-pot synthetic approach to the novel 5,6-dihydro-4H-[1,2,4]triazolo[4,3-alpha][1,5]benzodiazepines by thermal cyclization of 4-acylhydrazino-2,3-dihydro-IH-1,5-benzodiazepines is described.
引用
收藏
页码:943 / 948
页数:6
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