Microwave-assisted synthesis of phenylpyrimidine derivatives via Suzuki-Miyaura reactions in water

被引：13
|
作者：
Le, Yi [1 ,2 ,3 ]
Zhang, Yan [2 ]
Wang, Qin [2 ]
Rao, Nian [2 ]
Li, Dan [2 ]
Liu, Li [2 ,3 ]
Ouyang, Guiping [1 ,2 ,3 ]
Yan, Longjia [2 ,3 ]
机构：
[1] Guizhou Univ, Ctr Res & Dev Fine Chem,State Local Joint Lab Com, State Key Lab Breeding Base Green Pesticide & Agr, Key Lab Green Pesticide & Agr Bioengn,Minist Educ, Guiyang 550025, Peoples R China
[2] Guizhou Univ, Sch Pharmaceut Sci, Guiyang 550025, Peoples R China
[3] Guizhou Univ, Guizhou Engn Lab Synthet Drugs, Guiyang 550025, Peoples R China
来源：
TETRAHEDRON LETTERS | 2021年 / 68卷
关键词：
Phenylpyrimidine; Microwave; Suzuki-Miyaura; Water; Biguanidine;
D O I：
10.1016/j.tetlet.2021.152903
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient method was developed to prepare biphenylpyrimidine scaffolds via a Suzuki-Miyaura coupling reaction. In this procedure, the products were synthesized under microwave irradiation in water and analogues of biguanidine were employed as ligands. (C) 2021 Elsevier Ltd. All rights reserved.
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页数：4
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