Discovery and characterization of RLY-2608: The first allosteric, mutant, and isoform-selective inhibitor of PI3Kα

被引:4
|
作者
Pazolli, Ermira
Kipp, Randy
Boezio, Alessandro
Gunaydin, Hakan
Iskandar, Amanda
Zubrowski, Matthew
Williams, Bret
Shortsleeves, Kelley
Larivee, Alexandre
McLean, Tom
Michelsen, Klaus
Zeng, Hongtao
LaRochelle, Jonathan
Manna, Joe
DiPietro, Lucian
Mader, Mary
Bennet, Bindu
Wilbur, Jeremy
Wang, Qi
Pierce, Levi
Martin, Iain
Watters, James
Fortin, Pascal
Bergstrom, Donald
机构
关键词
D O I
10.1158/1535-7163.TARG-21-P251
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
P251
引用
收藏
页数:3
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