Cyclopropylboronic acid: synthesis and Suzuki cross-coupling reactions

被引：75
|
作者：
Wallace, DJ [1 ]
Chen, CY [1 ]
机构：
[1] Merck Res Labs, Dept Proc Res, Rahway, NJ 07065 USA
来源：
TETRAHEDRON LETTERS | 2002年 / 43卷 / 39期
关键词：
cyclopropylboronic acid; Suzuki cross-coupling; pharmaceutically acitve molecules;
D O I：
10.1016/S0040-4039(02)01606-4
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
An efficient synthesis of cyclopropylboronic acid is reported. This compound undergoes efficient Suzuki-type coupling reactions with a range of aryl and heteroarybromides. (C) 2002 Elsevier Science Ltd. All rights reserved.
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页码：6987 / 6990
页数：4
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