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- [31] Selective inhibition of FLT3 by gilteritinib in relapsed or refractory acute myeloid leukaemia: a multicentre, first-in-human, open-label, phase 1-2 studyLANCET ONCOLOGY, 2017, 18 (08): : 1061 - 1075Perl, Alexander E.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAAltman, Jessica K.论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Robert H Lurie Comprehens Canc Ctr, Chicago, IL 60611 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USACortes, Jorge论文数: 0 引用数: 0 h-index: 0机构: MD Anderson Canc Ctr, Houston, TX USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USASmith, Catherine论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Dept Leukemia, San Francisco, CA 94143 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USALitzow, Mark论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Rochester, MN USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USABaer, Maria R.论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Greenebaum Comprehens Canc Ctr, Baltimore, MD 21201 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAClaxton, David论文数: 0 引用数: 0 h-index: 0机构: Penn State Milton S Hershey Med Ctr, Hershey, PA USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAErba, Harry P.论文数: 0 引用数: 0 h-index: 0机构: Univ Alabama Birmingham, Dept Internal Med, Birmingham, AL USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAGill, Stan论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Global Dev, Northbrook, IL USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAGoldberg, Stuart论文数: 0 引用数: 0 h-index: 0机构: Hackensack Univ Med Ctr, Hackensack, NJ USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAJurcic, Joseph G.论文数: 0 引用数: 0 h-index: 0机构: Columbia Univ, Med Ctr, New York, NY USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USALarson, Richard A.论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Dept Med, Chicago, IL 60637 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USALiu, Chaofeng论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Global Dev, Northbrook, IL USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USARitchie, Ellen论文数: 0 引用数: 0 h-index: 0机构: Weill Cornell Med Coll, New York, NY USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USASchiller, Gary论文数: 0 引用数: 0 h-index: 0机构: Univ Calif Los Angeles, David Geffen Sch Med, Los Angeles, CA 90095 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USASpira, Alexander I.论文数: 0 引用数: 0 h-index: 0机构: Virginia Canc Specialists, Fairfax, VA USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAStrickland, Stephen A.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Ingram Canc Ctr, Nashville, TN 37208 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USATibes, Raoul论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Scottsdale, AZ USA Julius Maximilians Univ, Dept Internal Med, Wurzburg, Germany Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAUstun, Celalettin论文数: 0 引用数: 0 h-index: 0机构: Univ Minnesota, Dept Internal Med, Minneapolis, MN USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAWang, Eunice S.论文数: 0 引用数: 0 h-index: 0机构: Roswell Pk Canc Inst, Buffalo, NY 14263 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAStuart, Robert论文数: 0 引用数: 0 h-index: 0机构: Med Univ South Carolina, Hollings Canc Ctr, Charleston, SC 29425 USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USARoellig, Christoph论文数: 0 引用数: 0 h-index: 0机构: Univ Klinikum TU Dresden, Dept Internal Med, Dresden, Germany Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USANeubauer, Andreas论文数: 0 引用数: 0 h-index: 0机构: Univ Klinikum Giessen, Dept Internal Med, Marburg, Germany Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USAMartinelli, Giovanni论文数: 0 引用数: 0 h-index: 0机构: Univ Bologna, L & A Seragnoli, Bologna, Italy Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USABahceci, Erkut论文数: 0 引用数: 0 h-index: 0机构: Astellas Pharma Global Dev, Northbrook, IL USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USALevis, Mark论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Dept Oncol, Baltimore, MD USA Univ Penn, Abramson Comprehens Canc Ctr, Philadelphia, PA 19104 USA
- [32] First-in-human (FIH) phase I study of GST-HG161, a potent and highly selective c-met inhibitor, in patients with advanced solid tumor.JOURNAL OF CLINICAL ONCOLOGY, 2020, 38 (15)Li, Jin论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaGuo, Ye论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaXue, Junli论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaWu, Wenqiang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaChen, Shikui论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaTang, Yanan论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaXu, Xiongbin论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaLi, Gang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaHu, Lihong论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaLin, Yunfei论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaShen, Liang论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaXia, Yuanfeng论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaChan, Chi-Chung论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaWang, Zhouchong论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaNi, Dawen论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaDing, Charles论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R ChinaChen, Shuhui论文数: 0 引用数: 0 h-index: 0机构: Fudan Univ, Dept Med Oncol, Shanghai Canc Ctr, Shanghai, Peoples R China
- [33] CHIR258: A multitargeted growth factor receptor tyrosine kinase (RTK) inhibitor induces significant apoptosis of human FLT3 ITD acute myelogenous leukemia cells in vitro and in vivoBLOOD, 2004, 104 (11) : 496A - 496AMenezes, DL论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USAWiesmann, M论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USALee, SH论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USALee, I论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USAPeng, J论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USATang, Y论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USAYe, H论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USAOei, Y论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USAGoldbeck, C论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USAGarrett, EN论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USAHeise, C论文数: 0 引用数: 0 h-index: 0机构: Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA Chiron Corp, Biopharma R&D, Emeryville, CA 94608 USA
- [34] An open-label, single-dose, phase 1 study of the absorption, metabolism and excretion of quizartinib, a highly selective and potent FLT3 tyrosine kinase inhibitor, in healthy male subjects, for the treatment of acute myeloid leukemiaXENOBIOTICA, 2017, 47 (10) : 856 - 869Sanga, Madhu论文数: 0 引用数: 0 h-index: 0机构: Covance Labs Inc, Madison, WI USA Covance Labs Inc, Madison, WI USAJames, Joyce论文数: 0 引用数: 0 h-index: 0机构: Lyric Pharmaceut Inc, San Francisco, CA USA Covance Labs Inc, Madison, WI USAMarini, Joseph论文数: 0 引用数: 0 h-index: 0机构: Covance Labs Inc, Madison, WI USA Covance Labs Inc, Madison, WI USAGammon, Guy论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Inc, San Diego, CA 92121 USA Covance Labs Inc, Madison, WI USAHale, Christine论文数: 0 引用数: 0 h-index: 0机构: Covance Clin Res Unit, Madison, WI USA Covance Labs Inc, Madison, WI USALi, Jianke论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Inc, San Diego, CA 92121 USA Covance Labs Inc, Madison, WI USA
- [35] A first-in-human (FIH) phase I study of SAR12544, a novel selective MET kinase inhibitor, in patients (pts) with advanced solid tumors: Dose escalation resultsJOURNAL OF CLINICAL ONCOLOGY, 2014, 32 (15)Angevin, Eric论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, FranceSpitaleri, Gianluca论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, FranceHollebecque, Antoine论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, FranceDe Pas, Tommaso论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, FranceSoria, Jean-Charles论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, FranceHarnols, Marzia论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, FranceMazuir, Florent论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, FranceAssadourlan, Sylvie论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, FranceDe Marinis, Filippo论文数: 0 引用数: 0 h-index: 0机构: Inst Gustave Roussy, Villejuif, France
- [36] A Phase 1a/1b First in Human Study of PHI-101, a Potent Small Molecule Inhibitor of FLT3 in Relapsed and Refractory Acute Myeloid LeukemiaBLOOD, 2021, 138Yoon, Sung-Soo论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaShin, Dong-Yeop论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ Hosp, Dept Internal Med, Seoul, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaLee, Je-Hwan论文数: 0 引用数: 0 h-index: 0机构: Univ Ulsan, Coll Med, Asan Med Ctr, Dept Hematol, Seoul, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaJang, Jun Ho论文数: 0 引用数: 0 h-index: 0机构: Sungkyunkwan Univ, Sch Med, Samsung Med Ctr, Div Hematol Oncol,Dept Internal Med, Seoul, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaCheong, June-Won论文数: 0 引用数: 0 h-index: 0机构: Yonsei Univ, Severance Hosp, Coll Med, Dept Internal Med, Seoul, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaShin, Ho-Jin论文数: 0 引用数: 0 h-index: 0机构: Pusan Natl Univ Hosp, Dept Internal Med, Busan, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaLee, Jeong-Ok论文数: 0 引用数: 0 h-index: 0机构: Seoul Natl Univ, Bundang Hosp, Dept Internal Med, Seongnam, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaChoi, Yunsuk论文数: 0 引用数: 0 h-index: 0机构: Ulsan Univ Hosp, Dept Hematol & Oncol, Ulsan, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaPuliyayil, Anish论文数: 0 引用数: 0 h-index: 0机构: Albury Wodonga Canc Ctr, Border Med Oncol & Haematol, Albury, NSW, Australia Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaClarey, Joseph论文数: 0 引用数: 0 h-index: 0机构: ICON caner Ctr, N Mackay, Australia Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaJeejinlm论文数: 0 引用数: 0 h-index: 0机构: Pharos iBio Co Ltd, Anyang, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaNam, Ly-Youb论文数: 0 引用数: 0 h-index: 0机构: Pharos iBio Co Ltd, Anyang, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaKim, Kyu-Tae论文数: 0 引用数: 0 h-index: 0机构: Pharos iBio Co Ltd, Anyang, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaHan, June H-J.论文数: 0 引用数: 0 h-index: 0机构: Pharos iBio Co Ltd, Anyang, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaYoon, Jeong-Hyeok论文数: 0 引用数: 0 h-index: 0机构: Pharos iBio Co Ltd, Anyang, South Korea Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaNguyen, Bao论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Oncol, Baltimore, MD 21218 USA Albury Wodonga Canc Ctr, Border Med Oncol & Haematol, Albury, NSW, Australia Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaLi, Li论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Oncol, Baltimore, MD 21218 USA Albury Wodonga Canc Ctr, Border Med Oncol & Haematol, Albury, NSW, Australia Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South KoreaSmall, Donald论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Univ, Sch Med, Dept Oncol, Baltimore, MD 21218 USA Albury Wodonga Canc Ctr, Border Med Oncol & Haematol, Albury, NSW, Australia Seoul Natl Univ Hosp, Seoul Natl Univ Coll Med, Dept Internal Med, Seoul, South Korea
- [37] A first-in-human phase I study of SAR125844, a selective MET tyrosine kinase inhibitor, in patients with advanced solid tumours with MET amplificationEUROPEAN JOURNAL OF CANCER, 2017, 87 : 131 - 139Angevin, Eric论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, France Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceSpitaleri, Gianluca论文数: 0 引用数: 0 h-index: 0机构: Ist Europeo Oncol, Thorac Oncol Div, Via Ripamonti 435, I-20141 Milan, Italy Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceRodon, Jordi论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Barcelona, Vall dHebron Inst Oncol, Vall dHebron Univ Hosp, P Vall dHebron 119-129, Barcelona 08035, Spain Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceDotti, Katia论文数: 0 引用数: 0 h-index: 0机构: Ist Nazl Tumori, Via Venezian 1, I-20133 Milan, Italy Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceIsambert, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Ctr Georges Francois Leclerc, 1 Rue Prof Marion, F-21000 Dijon, France Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceSalvagni, Stefania论文数: 0 引用数: 0 h-index: 0机构: S Orsola Malpighi Univ Hosp Bologna, Oncol Med, Via Pietro Albertoni 15, I-40138 Bologna, Italy Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceMoreno, Victor论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ Fdn Jimenez Diaz, START MADRID FJD, Vda Reyes Catolicos 2, Madrid 28040, Spain Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceAssadourian, Sylvie论文数: 0 引用数: 0 h-index: 0机构: SANOFI, 54 Rue La Boetie, F-75008 Paris, France Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceGomez, Corinne论文数: 0 引用数: 0 h-index: 0机构: SANOFI, 54 Rue La Boetie, F-75008 Paris, France Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceHarnois, Marzia论文数: 0 引用数: 0 h-index: 0机构: SANOFI, 54 Rue La Boetie, F-75008 Paris, France Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceHollebecque, Antoine论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, France Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceAzaro, Analia论文数: 0 引用数: 0 h-index: 0机构: Univ Autonoma Barcelona, Vall dHebron Inst Oncol, Vall dHebron Univ Hosp, P Vall dHebron 119-129, Barcelona 08035, Spain Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceHervieu, Alice论文数: 0 引用数: 0 h-index: 0机构: Ctr Georges Francois Leclerc, 1 Rue Prof Marion, F-21000 Dijon, France Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceRihawi, Karim论文数: 0 引用数: 0 h-index: 0机构: S Orsola Malpighi Univ Hosp Bologna, Oncol Med, Via Pietro Albertoni 15, I-40138 Bologna, Italy Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, FranceDe Marinis, Filippo论文数: 0 引用数: 0 h-index: 0机构: Ist Europeo Oncol, Thorac Oncol Div, Via Ripamonti 435, I-20141 Milan, Italy Univ Paris Saclay, Gustave Roussy, DITEP, Drug Dev Dept, 114 Rue Edouard Vaillant, F-94805 Villejuif, France
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