Efficient synthesis of medium-sized cyclic amines by means of 2-nitrobenzenesulfonamide

被引：0
|
作者：
Kan, T [1 ]
Kobayashi, H [1 ]
Fukuyama, T [1 ]
机构：
[1] Univ Tokyo, Grad Sch Pharmaceut Sci, Bunkyo Ku, Tokyo 1130033, Japan
来源：
SYNLETT | 2002年 / 05期
关键词：
medium-sized cyclic amines; macrocyclization; 2-nitroberizenesulforiarnide; alkylation; Mitsunobu reaction;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Construction of medium-sized cyclic amines using 2-nitrobenzenesulfonamides is described, Under either conventional alkylation or Mitsunobu reaction conditions, the cyclization reaction proceeded efficiently to give eight- to ten-membered rings.
引用
收藏
页码：697 / 699
页数：3
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