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- [31] Triazoles as γ-secretase modulatorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (13) : 4083 - 4087Fischer, Christian论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAZultanski, Susan L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAZhou, Hua论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAMethot, Joey L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USABrown, W. Colby论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAMampreian, Dawn M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USASchell, Adam J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAShah, Sanjiv论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USANuthall, Hugh论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAHughes, Bethany L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USASmotrov, Nadja论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAKenific, Candia M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USACruz, Jonathan C.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAWalker, Deborah论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USABouthillette, Melanie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USANikov, George N.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USASavage, Dan F.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAJeliazkova-Mecheva, Valentina V.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USADiaz, Damaris论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USASzewczak, Alexander A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USABays, Nathan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAMiddleton, Richard E.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAMunoz, Benito论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USAShearman, Mark S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Boston, Boston, MA 02115 USA Merck Res Labs Boston, Boston, MA 02115 USA
- [32] Gamma-secretase modulators: a promising route for the treatment of Alzheimer's diseaseFRONTIERS IN MOLECULAR NEUROSCIENCE, 2023, 16Nordvall, Gunnar论文数: 0 引用数: 0 h-index: 0机构: AlzeCure Pharm AB, Huddinge, Sweden Karolinska Inst, Div Neurogeriatr, Ctr Alzheimer Res, Dept Neurobiol Care Sci & Soc, Stockholm, Sweden AlzeCure Pharm AB, Huddinge, SwedenLundkvist, Johan论文数: 0 引用数: 0 h-index: 0机构: AlzeCure Pharm AB, Huddinge, Sweden Karolinska Inst, Div Neurogeriatr, Ctr Alzheimer Res, Dept Neurobiol Care Sci & Soc, Stockholm, Sweden Sinfon Biotherapeut AB, Huddinge, Sweden AlzeCure Pharm AB, Huddinge, SwedenSandin, Johan论文数: 0 引用数: 0 h-index: 0机构: AlzeCure Pharm AB, Huddinge, Sweden Karolinska Inst, Div Neurogeriatr, Ctr Alzheimer Res, Dept Neurobiol Care Sci & Soc, Stockholm, Sweden AlzeCure Pharm AB, Huddinge, Sweden
- [33] Design and synthesis of novel methoxypyridine-derived gamma-secretase modulatorsBIOORGANIC & MEDICINAL CHEMISTRY, 2020, 28 (22)Rynearson, Kevin D.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USABuckle, Ronald N.论文数: 0 引用数: 0 h-index: 0机构: AMRI, Dept Med Chem, East Campus,3 Univ Pl, Rensselaer, NY 12144 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USAHerr, R. Jason论文数: 0 引用数: 0 h-index: 0机构: AMRI, Dept Med Chem, East Campus,3 Univ Pl, Rensselaer, NY 12144 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USAMayhew, Nicholas J.论文数: 0 引用数: 0 h-index: 0机构: AMRI, Dept Med Chem, East Campus,3 Univ Pl, Rensselaer, NY 12144 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USAChen, Xinchao论文数: 0 引用数: 0 h-index: 0机构: AMRI, Dept Med Chem, East Campus,3 Univ Pl, Rensselaer, NY 12144 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USAPaquette, William D.论文数: 0 引用数: 0 h-index: 0机构: AMRI, Dept Med Chem, East Campus,3 Univ Pl, Rensselaer, NY 12144 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USASakwa, Samuel A.论文数: 0 引用数: 0 h-index: 0机构: AMRI, Dept Med Chem, East Campus,3 Univ Pl, Rensselaer, NY 12144 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USAYang, Jinhai论文数: 0 引用数: 0 h-index: 0机构: AMRI, Dept Med Chem, East Campus,3 Univ Pl, Rensselaer, NY 12144 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USABarnes, Keith D.论文数: 0 引用数: 0 h-index: 0机构: AMRI, Dept Med Chem, East Campus,3 Univ Pl, Rensselaer, NY 12144 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USANguyen, Phuong论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USAMobley, William C.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USAJohnson, Graham论文数: 0 引用数: 0 h-index: 0机构: NuPharmAdvise, 3 Lakeside Dr, Sanbornton, NH 03269 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USALin, Juinn H.论文数: 0 引用数: 0 h-index: 0机构: Biopharm Consulting Partners, 2 Willet Dr, Ambler, PA 19002 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USATanzi, Rudolph E.论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Dept Neurol, Genet & Aging Res Unit, Charlestown, MA 02129 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USAWagner, Steven L.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USA Vet Adm San Diego Healthcare Syst, La Jolla, CA 92161 USA Univ Calif San Diego, Dept Neurosci, La Jolla, CA 92093 USA
- [34] γ-Secretase modulators exhibit selectivity for modulation of APP cleavage but inverse γ-secretase modulators do notALZHEIMERS RESEARCH & THERAPY, 2020, 12 (01)Lessard, Christian B.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA Univ Florida, Coll Med, McKnight Brain Inst, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USARodriguez, Edgardo论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Dept Pharmacol & Therapeut, McKnight Brain Inst, Ctr Translat Res Neurodegenerat Dis, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USALadd, Thomas B.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA Univ Florida, Coll Med, McKnight Brain Inst, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USAMinter, Lisa M.论文数: 0 引用数: 0 h-index: 0机构: Univ Massachusetts, Dept Vet & Anim Sci, Ctr Bioact Delivery, Inst Appl Life Sci, Amherst, MA 01003 USA Univ Massachusetts, Program Mol & Cellular Biol, Amherst, MA 01003 USA Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USAOsborne, Barbara A.论文数: 0 引用数: 0 h-index: 0机构: Univ Massachusetts, Dept Vet & Anim Sci, Ctr Bioact Delivery, Inst Appl Life Sci, Amherst, MA 01003 USA Univ Massachusetts, Program Mol & Cellular Biol, Amherst, MA 01003 USA Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA论文数: 引用数: h-index:机构:Golde, Todd E.论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA Univ Florida, Coll Med, McKnight Brain Inst, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USARan, Yong论文数: 0 引用数: 0 h-index: 0机构: Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA Univ Florida, Coll Med, McKnight Brain Inst, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA Univ Florida, Coll Med, Dept Neurosci & Neurol, Ctr Translat Res Neurodegenerat Dis, 1275 Ctr Dr,POB 100159, Gainesville, FL 32610 USA
- [35] γ-Secretase modulators exhibit selectivity for modulation of APP cleavage but inverse γ-secretase modulators do notAlzheimer's Research & Therapy, 12Christian B. Lessard论文数: 0 引用数: 0 h-index: 0机构: University of Florida,Department of Neuroscience and Neurology, Center for Translational Research in Neurodegenerative Disease, and McKnight Brain Institute, College of MedicineEdgardo Rodriguez论文数: 0 引用数: 0 h-index: 0机构: University of Florida,Department of Neuroscience and Neurology, Center for Translational Research in Neurodegenerative Disease, and McKnight Brain Institute, College of MedicineThomas B. Ladd论文数: 0 引用数: 0 h-index: 0机构: University of Florida,Department of Neuroscience and Neurology, Center for Translational Research in Neurodegenerative Disease, and McKnight Brain Institute, College of MedicineLisa M. Minter论文数: 0 引用数: 0 h-index: 0机构: University of Florida,Department of Neuroscience and Neurology, Center for Translational Research in Neurodegenerative Disease, and McKnight Brain Institute, College of MedicineBarbara A. Osborne论文数: 0 引用数: 0 h-index: 0机构: University of Florida,Department of Neuroscience and Neurology, Center for Translational Research in Neurodegenerative Disease, and McKnight Brain Institute, College of MedicineLucio Miele论文数: 0 引用数: 0 h-index: 0机构: University of Florida,Department of Neuroscience and Neurology, Center for Translational Research in Neurodegenerative Disease, and McKnight Brain Institute, College of MedicineTodd E. Golde论文数: 0 引用数: 0 h-index: 0机构: University of Florida,Department of Neuroscience and Neurology, Center for Translational Research in Neurodegenerative Disease, and McKnight Brain Institute, College of MedicineYong Ran论文数: 0 引用数: 0 h-index: 0机构: University of Florida,Department of Neuroscience and Neurology, Center for Translational Research in Neurodegenerative Disease, and McKnight Brain Institute, College of Medicine
- [36] Discovery of novel triazolobenzazepinones as γ-secretase modulators with central Aβ42 lowering in rodents and rhesus monkeysBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (17) : 3488 - 3494Fischer, Christian论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAZultanski, Susan L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAZhou, Hua论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAMethot, Joey L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAShah, Sanjiv论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAHayashi, Ikuo论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAHughes, Bethany L.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAMoxham, Christopher M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USABays, Nathan W.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USASmotrov, Nadya论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAHill, Armetta D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAPan, Bo-Sheng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAWu, Zhenhua论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAMoy, Lily Y.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USATanga, Flobert论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAKenific, Candia论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USACruz, Jonathan C.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAWalker, Deborah论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USABouthillette, Melanie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USANikov, George N.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USADeshmukh, Sujal V.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAJeliazkova-Mecheva, Valentina V.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USADiaz, Damaris论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAMichener, Maria S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA 19486 USA Merck Res Labs, Boston, MA 02115 USACook, Jacquelynn J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, West Point, PA 19486 USA Merck Res Labs, Boston, MA 02115 USAMunoz, Benito论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USAShearman, Mark S.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Boston, MA 02115 USA Merck Res Labs, Boston, MA 02115 USA
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