Synthesis of 3,4-dihydro-2H-pyrido[1,2-b]isoindol-1-one and 3,4-dihydro-2H-pyrido[1,2-b]pyrrolidin-1-one functionalized at the C-6 position by an intramolecular Horner-Wadsworth-Emmons reaction

被引：0

作者：

Gourves, JP ^{[1
]}

Couthon, H ^{[1
]}

Sturtz, G ^{[1
]}

机构：

[1] UFR Sci & Tech, Lab Chim Heteroorgan, F-29285 Brest, France

来源：

EUROPEAN JOURNAL OF ORGANIC CHEMISTRY | 1999年 / 1999卷 / 12期

关键词：

methylene-1,1-bisphosphonate; 3-bromoalkylimide; Horner-Wadsworth-Emmons reaction phosphonate complexes; heterocyclic compounds; cyclizations;

D O I：

10.1002/(SICI)1099-0690(199912)1999:12<3489::AID-EJOC3489>3.0.CO;2-F

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Novel polyheterocycles were prepared from a new annellation reaction which proceeds by nucleophilic substitution followed by an intramolecular Horner-Wads-worth-Emmons reaction between imides and beta-functionalized phosphonates.

引用

页码：3489 / 3493

页数：5

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