Extension of the SAR in the 1,2-diaminocyclohexane phenylacetamide template

被引：0
|
作者：
Zhao, SK [1 ]
Mizsak, SA [1 ]
Freeman, JP [1 ]
Szmuszkovicz, J [1 ]
机构：
[1] Univ Notre Dame, Dept Chem & Biochem, Notre Dame, IN 46556 USA
来源：
HETEROCYCLES | 2002年 / 58卷
关键词：
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Rigid analogs of 3,4-dichloro-N-methyl-N-[(1-methyl-2-piperidinyl)phenylmethyl]-benzeneacetamide (3), were prepared and allowed to extend the SAR of the U-50,488 template.
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页码：153 / 157
页数：5
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