Synthesis of a 5-substituted benzo[b]thiophene

被引：0

作者：

Wayne, GS ^{[1
]}

Lannoye, GS ^{[1
]}

Haight, AR ^{[1
]}

Parekh, SI ^{[1
]}

Zhang, WJ ^{[1
]}

Copp, RR ^{[1
]}

机构：

[1] Abbott Labs, Chem Proc Res, N Chicago, IL 60064 USA

来源：

HETEROCYCLES | 2000年 / 53卷 / 05期

关键词：

dimerci/benzo[b]thiophene; zileuton purity; Newman-Kwart rearrangement; regioselective Friedel-Crafts alkylation;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The synthesis of a 5-substituted dimeric benzo[b]thiophene (3), utilizing a Friedel-Crafts alkylation and subsequent Newman-Kwart rearrangement, is described.

引用

页码：1175 / +

页数：9

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