Synthesis of a 5-substituted benzo[b]thiophene

被引：0
|
作者：
Wayne, GS [1 ]
Lannoye, GS [1 ]
Haight, AR [1 ]
Parekh, SI [1 ]
Zhang, WJ [1 ]
Copp, RR [1 ]
机构：
[1] Abbott Labs, Chem Proc Res, N Chicago, IL 60064 USA
来源：
HETEROCYCLES | 2000年 / 53卷 / 05期
关键词：
dimerci/benzo[b]thiophene; zileuton purity; Newman-Kwart rearrangement; regioselective Friedel-Crafts alkylation;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The synthesis of a 5-substituted dimeric benzo[b]thiophene (3), utilizing a Friedel-Crafts alkylation and subsequent Newman-Kwart rearrangement, is described.
引用
收藏
页码：1175 / +
页数：9
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