A synthesis and transformations of alkyl 2-[2-cyano-2-(2-pyridinyl)ethenyl]amino-3-dimethylaminopropenoates.: A one-pot synthesis of pyrrolo[3,2-d]pyrimidin-4-ones

被引：0

作者：

Jukic, L ^{[1
]}

Svete, J ^{[1
]}

Golobic, A ^{[1
]}

Golic, L ^{[1
]}

Stanovnik, B ^{[1
]}

机构：

[1] Univ Ljubljana, Fac Chem & Chem Technol, Ljubljana 1000, Slovenia

来源：

HETEROCYCLES | 2000年 / 53卷 / 04期

关键词：

2-[2-cyano-2-(2-pyridinyl)ethenyl]amino-3-aminopropenoate; 4-pyridinyl-3-(2-aminovinyl)aminopyrrole;

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Alkyl 2-[2-cyano-2-(2-pyridinyl)ethenyl]amino-3-dimethylaminopropenoates (8) and (9) were transformed by heating into alkyl 2-[2-cyano-2-(2-pyridinyl)ethenyl]amino-3-[2-methoxycabonyl-4-(2-pyridinyl)-1H-pyrrol-3-yl]aminopropenoates (12) and (13). Compounds (8) and (9) can be transformed in the presence of primary aliphatic amines into substituted pyrrolo[3,2-d]pyrimidines (17-19).

引用

页码：805 / 820

页数：16

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