DETERMINANTS FOR PRODOMAIN INHIBITION OF THE TNF-α CONVERTING ENZYME (TACE) ZYMOGEN STATE

被引：0
|
作者：
Milla, Marcos E. [1 ]
机构：
[1] Roche, Palo Alto, CA 94304 USA
来源：
ADVANCES IN TNF FAMILY RESEARCH | 2011年 / 691卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：719 / 720
页数：2
相关论文
共 50 条
  • [1] TNF-α converting enzyme (TACE) as a therapeutic target
    Skotnicki, JS
    Levin, JI
    [J]. ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 38, 2003, 38 : 153 - 162
  • [2] Investigation of the Role of TNF-α Converting Enzyme (TACE) in the Inhibition of Cell Surface and Soluble TNF-α Production by Acute Ethanol Exposure
    von Maltzan, Kristine
    Tan, Wei
    Pruett, Stephen B.
    [J]. PLOS ONE, 2012, 7 (02):
  • [3] TNF-α converting enzyme (TACE) is inhibited by TIMP-3
    Amour, A
    Slocombe, PM
    Webster, A
    Butler, M
    Knight, CG
    Smith, BJ
    Stephens, PE
    Shelley, C
    Hutton, M
    Knäuper, V
    Docherty, AJP
    Murphy, G
    [J]. FEBS LETTERS, 1998, 435 (01) : 39 - 44
  • [4] Adamalysins -: A family of metzincins including TNF-α converting enzyme (TACE)
    Killar, L
    White, J
    Black, R
    Peschon, J
    [J]. INHIBITION OF MATRIX METALLOPROTEINASES: THERAPEUTIC APPLICATIONS, 1999, 878 : 442 - 452
  • [5] TNF-α-converting enzyme (TACE) expression in human and rat tissue.
    Knabb, MT
    Solomon, KA
    Reilly, TM
    Corjay, MH
    [J]. FASEB JOURNAL, 1999, 13 (04): : A204 - A204
  • [6] Chaperone-like properties of the prodomain of TNFα-converting enzyme (TACE) and the functional role of its cysteine switch
    Leonard, JD
    Lin, F
    Milla, ME
    [J]. BIOCHEMICAL JOURNAL, 2005, 387 : 797 - 805
  • [7] The discovery of novel tartrate-based TNF-α converting enzyme (TACE) inhibitors
    Rosner, Kristin E.
    Guo, Zhuyan
    Orth, Peter
    Shipps, Gerald W., Jr.
    Belanger, David B.
    Chan, Tin Yau
    Curran, Patrick J.
    Dai, Chaoyang
    Deng, Yongqi
    Girijavallabhan, Vinay M.
    Hong, Liwu
    Lavey, Brian J.
    Lee, Joe F.
    Li, Dansu
    Liu, Zhidan
    Popovici-Muller, Janeta
    Ting, Pauline C.
    Vaccaro, Henry
    Wang, Li
    Wang, Tong
    Yu, Wensheng
    Zhou, Guowei
    Niu, Xiaoda
    Sun, Jing
    Kozlowski, Joseph A.
    Lundell, Daniel J.
    Madison, Vincent
    McKittrick, Brian
    Piwinski, John J.
    Shih, Neng -Yang
    Siddiqui, M. Arshad
    Strickland, Corey O.
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (03) : 1189 - 1193
  • [8] Synthesis of piperidine phenyl sulfone hydroxamates as TACE (TNF-α converting enzyme) inhibitors
    Park, K
    Levin, JI
    Aplasca, A
    Du, ML
    Lovering, FE
    Condon, JS
    Zhang, YH
    Sun, LH
    Zhu, Y
    Xu, WX
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U151 - U152
  • [9] Novel TNF-α converting enzyme (TACE) inhibitors as potential treatment for inflammatory diseases
    Girijavallabhan, Vinay M.
    Chen, Lei
    Dai, Chaoyang
    Feltz, Robert J.
    Firmansjah, Luke
    Li, Dansu
    Kim, Seong Heon
    Kozlowski, Joseph A.
    Lavey, Brian J.
    Kosinski, Aneta
    Piwinski, John J.
    Popovici-Muller, Janeta
    Rizvi, Razia
    Rosner, Kristin E.
    Shankar, Banderpalle B.
    Shih, Neng-Yang
    Siddiqui, M. Arshad
    Tong, Ling
    Wong, Michael K. C.
    Yang, De-yi
    Yang, Liping
    Yu, Wensheng
    Zhou, Guowei
    Guo, Zhuyan
    Orth, Peter
    Madison, Vincent
    Bian, Hong
    Lundell, Daniel
    Niu, Xiaoda
    Shah, Himanshu
    Sun, Jing
    Umland, Shelby
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (24) : 7283 - 7287
  • [10] The mechanism by which cannabidiol (CBD) suppresses TNF-α secretion involves inappropriate localization of TNF-α converting enzyme (TACE)
    Frodella, Christa M.
    Liu, Liyuan
    Tan, Wei
    Pruett, Stephen B.
    Kaplan, Barbara L. F.
    [J]. CELLULAR IMMUNOLOGY, 2024, 397
12345