TNF-α converting enzyme (TACE) as a therapeutic target

被引:34
|
作者
Skotnicki, JS [1 ]
Levin, JI [1 ]
机构
[1] Wyeth Ayerst Res, Pearl River, NY 10965 USA
关键词
D O I
10.1016/S0065-7743(03)38017-0
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:153 / 162
页数:10
相关论文
共 50 条
  • [1] TNF-α converting enzyme (TACE) is inhibited by TIMP-3
    Amour, A
    Slocombe, PM
    Webster, A
    Butler, M
    Knight, CG
    Smith, BJ
    Stephens, PE
    Shelley, C
    Hutton, M
    Knäuper, V
    Docherty, AJP
    Murphy, G
    [J]. FEBS LETTERS, 1998, 435 (01) : 39 - 44
  • [2] Adamalysins -: A family of metzincins including TNF-α converting enzyme (TACE)
    Killar, L
    White, J
    Black, R
    Peschon, J
    [J]. INHIBITION OF MATRIX METALLOPROTEINASES: THERAPEUTIC APPLICATIONS, 1999, 878 : 442 - 452
  • [3] TNF-α-converting enzyme (TACE) expression in human and rat tissue.
    Knabb, MT
    Solomon, KA
    Reilly, TM
    Corjay, MH
    [J]. FASEB JOURNAL, 1999, 13 (04): : A204 - A204
  • [4] DETERMINANTS FOR PRODOMAIN INHIBITION OF THE TNF-α CONVERTING ENZYME (TACE) ZYMOGEN STATE
    Milla, Marcos E.
    [J]. ADVANCES IN TNF FAMILY RESEARCH, 2011, 691 : 719 - 720
  • [5] The discovery of novel tartrate-based TNF-α converting enzyme (TACE) inhibitors
    Rosner, Kristin E.
    Guo, Zhuyan
    Orth, Peter
    Shipps, Gerald W., Jr.
    Belanger, David B.
    Chan, Tin Yau
    Curran, Patrick J.
    Dai, Chaoyang
    Deng, Yongqi
    Girijavallabhan, Vinay M.
    Hong, Liwu
    Lavey, Brian J.
    Lee, Joe F.
    Li, Dansu
    Liu, Zhidan
    Popovici-Muller, Janeta
    Ting, Pauline C.
    Vaccaro, Henry
    Wang, Li
    Wang, Tong
    Yu, Wensheng
    Zhou, Guowei
    Niu, Xiaoda
    Sun, Jing
    Kozlowski, Joseph A.
    Lundell, Daniel J.
    Madison, Vincent
    McKittrick, Brian
    Piwinski, John J.
    Shih, Neng -Yang
    Siddiqui, M. Arshad
    Strickland, Corey O.
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (03) : 1189 - 1193
  • [6] Synthesis of piperidine phenyl sulfone hydroxamates as TACE (TNF-α converting enzyme) inhibitors
    Park, K
    Levin, JI
    Aplasca, A
    Du, ML
    Lovering, FE
    Condon, JS
    Zhang, YH
    Sun, LH
    Zhu, Y
    Xu, WX
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U151 - U152
  • [7] Novel TNF-α converting enzyme (TACE) inhibitors as potential treatment for inflammatory diseases
    Girijavallabhan, Vinay M.
    Chen, Lei
    Dai, Chaoyang
    Feltz, Robert J.
    Firmansjah, Luke
    Li, Dansu
    Kim, Seong Heon
    Kozlowski, Joseph A.
    Lavey, Brian J.
    Kosinski, Aneta
    Piwinski, John J.
    Popovici-Muller, Janeta
    Rizvi, Razia
    Rosner, Kristin E.
    Shankar, Banderpalle B.
    Shih, Neng-Yang
    Siddiqui, M. Arshad
    Tong, Ling
    Wong, Michael K. C.
    Yang, De-yi
    Yang, Liping
    Yu, Wensheng
    Zhou, Guowei
    Guo, Zhuyan
    Orth, Peter
    Madison, Vincent
    Bian, Hong
    Lundell, Daniel
    Niu, Xiaoda
    Shah, Himanshu
    Sun, Jing
    Umland, Shelby
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (24) : 7283 - 7287
  • [8] The mechanism by which cannabidiol (CBD) suppresses TNF-α secretion involves inappropriate localization of TNF-α converting enzyme (TACE)
    Frodella, Christa M.
    Liu, Liyuan
    Tan, Wei
    Pruett, Stephen B.
    Kaplan, Barbara L. F.
    [J]. CELLULAR IMMUNOLOGY, 2024, 397
  • [9] TNF-α converting enzyme (TACE) protein expression in different clinical subtypes of multiple sclerosis
    Comabella, Manuel
    Romera, Cristina
    Camina, Montse
    Perkal, Hector
    Moro, Maria A.
    Leza, Juan C.
    Lizasoain, Ignacio
    Castillo, Mireia
    Montalban, Xavier
    [J]. JOURNAL OF NEUROLOGY, 2006, 253 (06) : 701 - 706
  • [10] Design, synthesis and evaluation of β-benzamido hydroxamic acid inhibitors of TNF-α converting enzyme (TACE).
    Ott, GR
    Lu, ZH
    Asakawa, N
    Covington, MB
    Qian, MX
    Liu, RQ
    Newton, RC
    Christ, DD
    Decicco, CP
    Duan, JJW
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2004, 228 : U966 - U966