Synthesis and antibacterial screening of N-sulphonamoylphenylamino-3-chloro-4-phenylazetidin-2-ones

被引：0
|
作者：
Sharma, P [1 ]
Indapurkar, P [1 ]
Mandloi, A [1 ]
机构：
[1] Devi Ahilya Univ, Inst Chem Sci, Indore 452001, Madhya Pradesh, India
来源：
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 1998年 / 37卷 / 05期
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D O I：
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中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Some new N-sulphonamoylphenylamino-3-chloro-4-phenylazetidin-2-ones 2a-f have been synthesised and their structures have been established on the basis of their elemental, IR, and H-1 NMR data. Compounds 2a-f show significant antibacterial activity. 1-[4'(5 "-6'-dimethoxypyrimidinosulphonamoyl) phenylamino]-3 -chloro-4-phenylazetidin-2-one 2e has been found to be more potent antibacterial agent against E. coli.
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页码：521 / 522
页数：2
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