Synthesis of [18F]fluoromethyl-PBR28-d2 and its preclinical comparison with [18F] fluoromethyl-PBR28 in a rat model of neuroinflammation

被引：0
|
作者：
Moon, Byung Seok [1 ]
Jung, Jae Ho [1 ]
Park, Hyun Soo [2 ]
Contino, Marialessandra [3 ]
Denora, Nunzio [3 ]
Lee, Byung Chul [1 ]
Kim, Sang Eun [2 ]
机构：
[1] Seoul Natl Univ, Coll Med, Bundang Hosp, Dept Nucl Med, Seoul, South Korea
[2] Seoul Natl Univ, Grad Sch Convergence Sci & Technol, Dept Transdisciplinary Studies, Seoul, South Korea
[3] Univ Bari A Moro, Dept Pharm Drug Sci, Bari, Italy
来源：
JOURNAL OF NUCLEAR MEDICINE | 2015年 / 56卷 / 03期
关键词：
D O I：
暂无
中图分类号：
R8 [特种医学]; R445 [影像诊断学];
学科分类号：
1002 ; 100207 ; 1009 ;
摘要：
1089
引用
收藏
页数：1
相关论文
共 50 条
  • [21] Facile automated synthesis of [18F]fluoromethyl-d2 group in a commercial 18F-synthetic module
    Jo, Byeong Min
    Moon, Byung Seok
    Lee, Hong Jin
    Park, Hyun Sik
    Lee, Byung Chul
    Kim, Sang Eun
    [J]. JOURNAL OF NUCLEAR MEDICINE, 2015, 56 (03)
  • [22] Improved synthesis of [18F]fluoromethyl tosylate, a convenient reagent for radiofluoromethylations
    Neal, TR
    Apana, S
    Berridge, MS
    [J]. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2005, 48 (08): : 557 - 568
  • [23] Automated HPLC free microfluidic synthesis of [18F]fluoromethyl tosylate
    Winkle, Richard F.
    Smith, Graham
    de Mello, Andrew J.
    Aboagye, Eric O.
    [J]. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2011, 54 : S544 - S544
  • [24] Direct Comparison of [18F]F-DPA with [18F]DPA-714 and [11C]PBR28 for Neuroinflammation Imaging in the same Alzheimer’s Disease Model Mice and Healthy Controls
    Francisco R. López-Picón
    Thomas Keller
    Diana Bocancea
    Jatta S. Helin
    Anna Krzyczmonik
    Semi Helin
    Annelaure Damont
    Frédéric Dollé
    Juha O. Rinne
    Merja Haaparanta-Solin
    Olof Solin
    [J]. Molecular Imaging and Biology, 2022, 24 : 157 - 166
  • [25] Automated production of [18F]PBR111 for imaging neuroinflammation in humans
    Onega, Mayca
    Barletta, Julien
    Pampols-Maso, Sabina
    Singleton, Goerkem
    Passchier, Jan
    Bennacef, Idriss
    [J]. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2011, 54 : S440 - S440
  • [26] Synthesis of 6-[18F]fluoro-PBR28, a novel radiotracer for imaging the TSPO 18 kDa with PET
    Damont, Annelaure
    Boisgard, Raphael
    Kuhnast, Bertrand
    Lemee, Frederic
    Raggiri, Guillaume
    Scarf, Alana M.
    Da Pozzo, Eleonora
    Selleri, Silvia
    Martini, Claudia
    Tavitian, Bertrand
    Kassiou, Michael
    Dolle, Frederic
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (16) : 4819 - 4822
  • [27] [18F]PBR146 and [18F]DPA-714 in vivo Imaging of Neuroinflammation in Chronic Hepatic Encephalopathy Rats
    Kong, Xiang
    Luo, Song
    Wang, Yun Fei
    Yang, Gui Fen
    Lu, Guang Ming
    Zhang, Long Jiang
    [J]. FRONTIERS IN NEUROSCIENCE, 2021, 15
  • [28] TSPO PET ligands [18F]PBR06 and [18F]DPA-714 for glioma imaging: A preclinical comparison of kinetic parameters
    Tantawy, Mohammed
    Tang, Dewei
    Buck, Jason
    Manning, H. Charles
    [J]. JOURNAL OF NUCLEAR MEDICINE, 2011, 52
  • [29] Evaluation of [18F]PBR111 in a rat model of neuroinflammation: A new radiotracer for the TSPO 18 kDa (peripheral benzodiazepine receptor)
    Van Camp, Nadja
    Chauveau, Fabien
    Boisgard, Raphael
    Jego, Benoit
    Siquier, Karine
    Kuhnast, Bertrand
    Gregoire, Marie Claude
    Katsifis, Andrew
    Dolle, Frederic
    Tavitian, Bertrand
    [J]. JOURNAL OF NUCLEAR MEDICINE, 2009, 50
  • [30] Synthesis of 4-([18F]fluoromethyl)-2-chlorophenylisothiocyanate:: A novel bifunctional 18F-labelling agent
    Wüst, F
    Müller, M
    Bergmann, R
    [J]. RADIOCHIMICA ACTA, 2004, 92 (4-6) : 349 - 353
12345