Expeditious preparation of aristeromycin analogues.: Synthesis of 2′,3′-dideoxyaristeromycin

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作者
Comin, MJ [1 ]
Rodriguez, JB [1 ]
机构
[1] Univ Buenos Aires, Fac Ciencias Exactas & Nat, Dept Quim Organ, RA-1428 Buenos Aires, DF, Argentina
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O6 [化学];
学科分类号
0703 ;
摘要
The preparation of the carbocyclic nucleoside 2',3'dideoxyaristeromycin was carried out in ten steps starting from the readily available cyclohex-2-enone. A convergent approach was envisioned using a Mitsunobu metholology as key step to incorporate the heterocyclic base onto the carbocyclic ring.
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页码:131 / 138
页数:8
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