Juvenile hormone activity of ethyl 4-(2-aryloxyhexyloxy)benzoates with precocious metamorphosis-inducing activity

被引：1

作者：

Fujita, Norihiro

Ashibe, Kiyo

Yamada, Naotaka

Shiotsuki, Takahiro

Kiuchi, Makoto

Kuwano, Eiichi ^{[1
]}

机构：

[1] Kyushu Univ, Fac Agr, Dept Appl Genet & Pest Management, Lab Pesticide Chem, Fukuoka 812, Japan

[2] Natl Inst Agrobiol Sci, Invertebrate Gene Funct Res Unit, Tsukuba 305, Japan

来源：

BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY | 2007年 / 71卷 / 09期

关键词：

juvenile hormone; precocious metamorphosis; anti-juvenile hormone; silkworm;

D O I：

10.1271/bbb.70265

中图分类号：

Q5 [生物化学]; Q7 [分子生物学];

学科分类号：

071010 ; 081704 ;

摘要：

Ethyl 4-[2-(6-methyl-3-pyridyloxy)hexyloxy]benzoate (1) and ethyl 4-(2-phenoxyhexyloxy)benzoate (2), which induce precocious metamorphosis in larvae of Bombyx mori, a clear sign of juvenile hormone (JH) deficiency, showed JH activity when topically applied to allatectomized 4th instar larvae of B. mori. Compounds 1 and 2 induced precocious metamorphosis with doses at which they were effective as JH agonists.

引用

页码：2333 / 2334

页数：2

共 50 条

[11] Ethyl 4-[(1-substituted indol-2-yl)methoxy]benzoates and indoline derivatives: Anti-juvenile hormone and juvenile hormone activities
Furuta, Kenjiro
Yoshida, Shuhei
Fujita, Norihiro
Yamada, Naotaka
Kuwano, Eiichi
JOURNAL OF PESTICIDE SCIENCE, 2009, 34 (03) : 177 - 180
[12] Anti-juvenile hormone activity of ethyl 4-[(7-substituted 1,4-benzodioxan-6-yl)methyl]benzoates and their effect on the juvenile hormone titer in the hemolymph of the silkworm, Bombyx mori
Yamada, Naoko
Maeda, Kei
Masumoto, Masaaki
Inagaki, Yoshitaka
Furuta, Kenjiro
JOURNAL OF PESTICIDE SCIENCE, 2016, 41 (02) : 38 - 43
[13] Analgesic Activity of Ethyl 4-(6-Aryl-5-Benzoyl-4-Hydroxy-2-Thioxohexahydropyrimidine-4-Carboxamido)Benzoates
Zamaraeva, T. M.
Gorgopina, E. V.
PHARMACEUTICAL CHEMISTRY JOURNAL, 2025, : 1694 - 1696
[14] Synthesis and anti-juvenile hormone activity of ethyl 4-[2-(6-methyl-3-pyridyloxy)alkyloxylbenzoates
Fujita, N
Furuta, K
Shirahashi, H
Hong, S
Shiotsuki, T
Kuwano, E
JOURNAL OF PESTICIDE SCIENCE, 2005, 30 (03) : 192 - 198
[15] Synthesis and Analgesic Activity of Etyl 4-[(4-Aryl-2-hydroxy-4-oxobut-2-enoyl)amino]benzoates
Gein, V. L.
Romanova, A. V.
Bobrovskaya, O. V.
Nazarets, O. V.
Makhmudov, R. R.
Gradova, E. V.
RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2022, 92 (11) : 2231 - 2234
[16] Synthesis and Analgesic Activity of Etyl 4-[(4-Aryl-2-hydroxy-4-oxobut-2-enoyl)amino]benzoates
V. L. Gein
A. V. Romanova
O. V. Bobrovskaya
O. V. Nazarets
R. R. Makhmudov
Е. V. Gradova
Russian Journal of General Chemistry, 2022, 92 : 2231 - 2234
[17] COMPOUNDS WITH INSECT JUVENILE HORMONE-ACTIVITY .2. SYNTHESIS OF 4-OXAFARNESANE INSECT JUVENILE HORMONE MIMICS
PATIL, MM
PATWARDHAN, SA
GUPTA, AS
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1978, 16 (07): : 625 - 627
[18] An anti-juvenile hormone agent, ethyl 4-(2-benzylhexyloxy)benzoate, inhibits juvenile hormone synthesis through the suppression of the transcription of juvenile hormone biosynthetic enzymes in the corpora allata in Bombyx mori
Kaneko, Yu
Furuta, Kenjiro
Kuwano, Eiichi
Hiruma, Kiyoshi
INSECT BIOCHEMISTRY AND MOLECULAR BIOLOGY, 2011, 41 (10) : 788 - 794
[19] Synthesis and Cardiotropic Activity of 1-(Methoxybenzyl)-4-{2-[(Methoxybenzyl)-Amino]Ethyl}Piperazines
G. V. Mokrov
A. M. Likhosherstov
V. V. Barchukov
V. N. Stolyaruk
I. B. Tsorin
M. B. Vititnova
A. G. Rebeko
S. A. Kryzhanovskii
T. A. Gudasheva
Pharmaceutical Chemistry Journal, 2019, 53 : 786 - 791
[20] Synthesis and Cardiotropic Activity of 1-(Methoxybenzyl)-4-{2-[(Methoxybenzyl)-Amino]Ethyl}Piperazines
Mokrov, G. V.
Likhosherstov, A. M.
Barchukov, V. V.
Stolyaruk, V. N.
Tsorin, I. B.
Vititnova, M. B.
Rebeko, A. G.
Kryzhanovskii, S. A.
Gudasheva, T. A.
PHARMACEUTICAL CHEMISTRY JOURNAL, 2019, 53 (09) : 786 - 791

← 1 2 3 4 5 →