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- [21] Hurdles in the Drug Discovery of Cathepsin K InhibitorsCURRENT TOPICS IN MEDICINAL CHEMISTRY, 2010, 10 (07) : 733 - 744Kometani, Motohiko论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res Tsukuba, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res Tsukuba, Tsukuba, Ibaraki 3002611, JapanNonomura, Kazuhiko论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res Tsukuba, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res Tsukuba, Tsukuba, Ibaraki 3002611, JapanTomoo, Takashi论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res Tsukuba, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res Tsukuba, Tsukuba, Ibaraki 3002611, JapanNiwa, Satoru论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res Tsukuba, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res Tsukuba, Tsukuba, Ibaraki 3002611, Japan
- [22] Peptide ketobenzoxazole inhibitors bound to cathepsin KBIOCHEMISTRY, 2003, 42 (51) : 15018 - 15028McGrath, ME论文数: 0 引用数: 0 h-index: 0机构: Celera, San Francisco, CA USA Celera, San Francisco, CA USASprengeler, PA论文数: 0 引用数: 0 h-index: 0机构: Celera, San Francisco, CA USA Celera, San Francisco, CA USAHill, CM论文数: 0 引用数: 0 h-index: 0机构: Celera, San Francisco, CA USA Celera, San Francisco, CA USAMartichonok, V论文数: 0 引用数: 0 h-index: 0机构: Celera, San Francisco, CA USA Celera, San Francisco, CA USACheung, H论文数: 0 引用数: 0 h-index: 0机构: Celera, San Francisco, CA USA Celera, San Francisco, CA USASomoza, JR论文数: 0 引用数: 0 h-index: 0机构: Celera, San Francisco, CA USA Celera, San Francisco, CA USAPalmer, JT论文数: 0 引用数: 0 h-index: 0机构: Celera, San Francisco, CA USA Celera, San Francisco, CA USAJanc, JW论文数: 0 引用数: 0 h-index: 0机构: Celera, San Francisco, CA USA Celera, San Francisco, CA USA
- [23] Difluoroethylamines as an amide isostere in inhibitors of cathepsin KBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (03) : 920 - 923Isabel, Elise论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaMellon, Christophe论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaBoyd, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaChauret, Nathalie论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaDeschenes, Denis论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaDesmarais, Sylvie论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaFalgueyret, Jean-Pierre论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaGauthier, Jacques Yves论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaKhougaz, Karine论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaLau, Cheuk K.论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaLeger, Serge论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaLevorse, Dorothy A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmaceut Analyt Chem, Rahway, NJ 07065 USA Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaLi, Chun Sing论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaMasse, Frederic论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaPercival, M. David论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaRoy, Bruno论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaScheigetz, John论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaTherien, Michel论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaTruong, Vouy Linh论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaWesolowski, Gregg论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Bone Biol & Osteoporosis, West Point, PA 19486 USA Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaYoung, Robert N.论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaZamboni, Robert论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, CanadaBlack, W. Cameron论文数: 0 引用数: 0 h-index: 0机构: Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Quebec City, PQ H9H 3L1, Canada
- [24] Cathepsin K inhibitors, 2000-2004EXPERT OPINION ON THERAPEUTIC PATENTS, 2005, 15 (01) : 33 - 48Cai, JQ论文数: 0 引用数: 0 h-index: 0机构: Organon Res Labs Ltd, Dept Med Chem, Newhouse ML1 5SH, Scotland Organon Res Labs Ltd, Dept Med Chem, Newhouse ML1 5SH, ScotlandJamieson, C论文数: 0 引用数: 0 h-index: 0机构: Organon Res Labs Ltd, Dept Med Chem, Newhouse ML1 5SH, Scotland Organon Res Labs Ltd, Dept Med Chem, Newhouse ML1 5SH, ScotlandMoir, J论文数: 0 引用数: 0 h-index: 0机构: Organon Res Labs Ltd, Dept Med Chem, Newhouse ML1 5SH, Scotland Organon Res Labs Ltd, Dept Med Chem, Newhouse ML1 5SH, ScotlandRankovic, Z论文数: 0 引用数: 0 h-index: 0机构: Organon Res Labs Ltd, Dept Med Chem, Newhouse ML1 5SH, Scotland Organon Res Labs Ltd, Dept Med Chem, Newhouse ML1 5SH, Scotland
- [25] Development and evaluation of new cathepsin K inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241Tha, Soe论文数: 0 引用数: 0 h-index: 0机构: Western Illinois Univ, Dept Chem, Macomb, IL 61455 USA Western Illinois Univ, Dept Chem, Macomb, IL 61455 USALiang, Kenneth论文数: 0 引用数: 0 h-index: 0机构: Western Illinois Univ, Dept Chem, Macomb, IL 61455 USA Western Illinois Univ, Dept Chem, Macomb, IL 61455 USAObregon, Roxana论文数: 0 引用数: 0 h-index: 0机构: Western Illinois Univ, Dept Chem, Macomb, IL 61455 USA Western Illinois Univ, Dept Chem, Macomb, IL 61455 USAKadasala, Naveen Reddy论文数: 0 引用数: 0 h-index: 0机构: Western Illinois Univ, Dept Chem, Macomb, IL 61455 USA Western Illinois Univ, Dept Chem, Macomb, IL 61455 USAWen, Lisa论文数: 0 引用数: 0 h-index: 0机构: Western Illinois Univ, Dept Chem, Macomb, IL 61455 USA Western Illinois Univ, Dept Chem, Macomb, IL 61455 USAHuang, Jenq Kuen论文数: 0 引用数: 0 h-index: 0机构: Western Illinois Univ, Dept Chem, Macomb, IL 61455 USA Western Illinois Univ, Dept Chem, Macomb, IL 61455 USAMcConnell, Rose论文数: 0 引用数: 0 h-index: 0机构: Western Illinois Univ, Dept Chem, Macomb, IL 61455 USA Western Illinois Univ, Dept Chem, Macomb, IL 61455 USA
- [26] Thiosemicarbazones as potent and selective cathepsin K inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 241Chavarria, Gustavo E.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USADevanna, Kishore K. Gaddale论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAJones, Lindsay M.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAMacDonough, Matthew T.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAYoo, Grace K.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USALocke, Ashleigh论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USADeliz, Rafael论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAChaplin, David J.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USASiim, Bronwyn G.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAChen, Shen-En论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USAPinney, Kevin G.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USATrawick, Mary L.论文数: 0 引用数: 0 h-index: 0机构: Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA Baylor Univ, Dept Chem & Biochem, Waco, TX 76798 USA
- [27] New Synthetic Quinolines as Cathepsin K InhibitorsJOURNAL OF THE BRAZILIAN CHEMICAL SOCIETY, 2020, 31 (08) : 1605 - 1613Silva, Taynara L.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazil Fac Dent, 2350 Hlth Sci Mall, Vancouver, BC V6T 1Z3, Canada UBC Ctr Blood Res, 2350 Hlth Sci Mall, Vancouver, BC V6T 1Z3, Canada Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, BrazilBartolomeu, Aloisio de A.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazil Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazilde Jesus, Hugo C. R.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazil Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazilde Oliveira, Kleber T.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazil Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, BrazilFernandes, Joao B.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazil Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, BrazilBromme, Dieter论文数: 0 引用数: 0 h-index: 0机构: Fac Dent, 2350 Hlth Sci Mall, Vancouver, BC V6T 1Z3, Canada UBC Ctr Blood Res, 2350 Hlth Sci Mall, Vancouver, BC V6T 1Z3, Canada Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, BrazilVieira, Paulo C.论文数: 0 引用数: 0 h-index: 0机构: Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazil Univ Sao Paulo, Fac Ciencias Farmaceut Ribeirao Preto, BR-14040903 Ribeirao Preto, SP, Brazil Univ Fed Sao Carlos, Dept Quim, Km 235, BR-13565905 Sao Carlos, SP, Brazil
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- [29] Effect of cathepsin K inhibitors on bone resorptionJOURNAL OF MEDICINAL CHEMISTRY, 2008, 51 (17) : 5459 - 5462Teno, Naoki论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanMasuya, Keiichi论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanEhara, Takeru论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanKosaka, Takatoshi论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanMiyake, Takahiro论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanIrie, Osamu论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanHitomi, Yuko论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanMatsuura, Naoko论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanUmemura, Ichiro论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanIwasaki, Genji论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanFukaya, Hiroaki论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanToriyama, Kazuhiro论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanUchiyama, Noriko论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanNonomura, Kazuhiko论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanSugiyama, Ikuo论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, JapanKometani, Motohiko论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan Novartis Inst BioMed Res, Tsukuba, Ibaraki 3002611, Japan
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