SYNTHESIS AND ACTIVITY OF PHOSPHINIC TRIPEPTIDE ANALOGUES AS INHIBITORS OF CATHEPSIN C

被引：0
|
作者：
Mucha, A. [1 ]
Pawelczak, M. [2 ]
Kafarski, P. [1 ,2 ]
机构：
[1] Wroclaw Univ Technol, Inst Organ Chem Biochem & Biotechnol, PL-50370 Wroclaw, Poland
[2] Univ Opole, Inst Chem, Opole, Poland
来源：
JOURNAL OF PEPTIDE SCIENCE | 2004年 / 10卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：212 / 212
页数：1
相关论文
共 50 条
  • [41] Synthesis of imidazole phosphinic acids as I4AA analogues
    Orain, D
    Mattes, H
    TETRAHEDRON LETTERS, 2006, 47 (08) : 1253 - 1255
  • [42] Design and synthesis of dipeptidyl nitriles as potent, selective, and reversible inhibitors of cathepsin C
    Guay, Daniel
    Beaulieu, Christian
    Reddy, T. Jagadeeswar
    Zamboni, Robert
    Methot, Nathalie
    Rubin, Joel
    Ethier, Diane
    Percival, M. David
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (18) : 5392 - 5396
  • [43] Synthesis and antitumor activity of litseaone B analogues as tubulin polymerisation inhibitors
    Yang, Wei
    Peng, Huining
    Huang, Yong
    Peng, Zhiyun
    Wang, Guangcheng
    JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2022, 37 (01) : 2530 - 2539
  • [44] Triphenylethylene analogues: Design, synthesis and evaluation of antitumor activity and topoisomerase inhibitors
    Rani, Sudesh
    Paul, Kamaldeep
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2020, 208
  • [45] An efficient one-pot synthesis of bis(α-aminoalkyl)phosphinic acids, phosphorus-isosteric analogues of HIV protease inhibitors
    Vinyukov, Alexey V.
    Borodachev, Alexey V.
    Starikov, Andrey S.
    Afanasyev, Alexey V.
    Dmitriev, Maxim E.
    Lednev, Boris V.
    Ragulin, Valery V.
    MENDELEEV COMMUNICATIONS, 2018, 28 (03) : 295 - 296
  • [46] ANGIOTENSIN-CONVERTING ENZYME-INHIBITORS - SYNTHESIS AND BIOLOGICAL-ACTIVITY OF N-SUBSTITUTED TRIPEPTIDE INHIBITORS
    SAWAYAMA, T
    TSUKAMOTO, M
    SASAGAWA, T
    NISHIMURA, K
    DEGUCHI, T
    TAKEYAMA, K
    HOSOKI, K
    CHEMICAL & PHARMACEUTICAL BULLETIN, 1990, 38 (01) : 110 - 115
  • [47] C-4 analogues of podophyllotoxin as tubulin inhibitors: synthesis, biological evaluation, and structure-activity relationship
    Lu, Breanna
    Xu, Lexi
    Chen, Harriet
    Yu, Grace
    Khow, Kimberly
    Yang, Stella
    Dinker, Arushi
    Njoo, Edward
    NATURAL PRODUCT RESEARCH, 2024,
  • [48] Effects of α-melanotropin C-terminal tripeptide analogues on macrophage NO production
    Muceniece, R
    Krigere, L
    Süli-Vargha, H
    Wikberg, JES
    PEPTIDES, 2003, 24 (05) : 701 - 707
  • [49] Design and pharmacological activity of phosphinic acid based NAALADase inhibitors
    Jackson, PF
    Tays, KL
    Maclin, KM
    Ko, YS
    Li, WX
    Vitharana, D
    Tsukamoto, T
    Stoermer, D
    Lu, XCM
    Wozniak, K
    Slusher, BS
    JOURNAL OF MEDICINAL CHEMISTRY, 2001, 44 (24) : 4170 - 4175
  • [50] Role of cathepsin A and cathepsin C in the regulation of glycosidase activity
    Minarowska, Alina
    Minarowski, Lukasz
    Karwowska, Alicja
    Milewska, Anna Justyna
    Gacko, Marek
    FOLIA HISTOCHEMICA ET CYTOBIOLOGICA, 2012, 50 (01) : 20 - 24
12345