Selective reduction and functionalization of diethyl 1-alkyl-1H-indole-2,3-dicarboxylates

被引：12
|
作者：
Sayyed, Iliyas Ali [1 ]
Alex, Karolin [1 ]
Tillack, Annegret [1 ]
Schwarz, Nicolle [1 ]
Spannenberg, Anke [1 ]
Michalik, Dirk [1 ]
Beller, Matthias [1 ]
机构：
[1] Univ Rostock, Leibniz Inst Katalyse eV, D-18059 Rostock, Germany
来源：
TETRAHEDRON | 2008年 / 64卷 / 20期
关键词：
D O I：
10.1016/j.tet.2008.03.011
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A convenient and highly selective reduction of easily accessible indole-2,3-dicarboxylates is described. Ten different 1-alkyl-2-formyl-1H-indole-3-carboxylates are obtained in high yield and represent interesting building blocks for novel indoles. (C) 2008 Elsevier Ltd. All rights reserved.
引用
收藏
页码：4590 / 4595
页数：6
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