A Convenient Synthesis of Some New 1,3,4-Thiadiazoles, Thiazoles, Pyrazolo[1,5-a]pyrimidines, Pyrazolo[5,1-c]triazine, and Thieno[3,2-d]pyrimidines Containing 5-Bromobenzofuran Moiety

被引：8

作者：

Abdelhamid, Abdou O. ^{[1
]}

Fahmi, Abdelgawad A. ^{[1
]}

Baaiu, Basma S. ^{[1
]}

机构：

[1] Cairo Univ, Dept Chem, Fac Sci, Giza 12613, Egypt

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 2016年 / 53卷 / 04期

关键词：

HYDRAZONOYL HALIDES; ANTIMICROBIAL ACTIVITY; 5-ARYLAZOTHIAZOLES; DERIVATIVES; AGENTS;

D O I：

10.1002/jhet.2383

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

1,3,4-Thiadiazoles, pyrazolo[1,5-a]pyrimidines, pyrazolo[5,1-c]triazine, and thieno[3,2-d]pyrimidines were synthesized from 1-(5-bromobenzofuran-2-yl)ethanone. The structures of the newly synthesized compounds were elucidated by elemental analysis, spectral data, chemical transformation, and alternative synthesis route whenever possible.

引用

页码：1292 / 1303

页数：12

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