INTERINDIVIDUAL VARIABILITY IN CYP2D6 ACTIVITY IN HUMAN LIVER MICROSOMES TO CHARACTERIZE RARE GENETIC VARIATION.

被引:0
|
作者
Dalton, R. [1 ]
Phillips, B. [2 ]
Risler, L. [2 ]
Shen, D. D. [2 ]
Woodahl, E. L. [1 ]
机构
[1] Univ Montana, Missoula, MT 59812 USA
[2] Univ Washington, Seattle, WA 98195 USA
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
PII-023
引用
收藏
页码:S65 / S66
页数:2
相关论文
共 50 条
  • [21] INVOLVEMENT OF CYP2D6 IN OXIDATIVE-METABOLISM OF CINNARIZINE AND FLUNARIZINE IN HUMAN LIVER-MICROSOMES
    NARIMATSU, S
    KARIYA, S
    ISOZAKI, S
    OHMORI, S
    KITADA, M
    HOSOKAWA, S
    MASUBUCHI, Y
    SUZUKI, T
    BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1993, 193 (03) : 1262 - 1268
  • [22] How and Why to Screen for CYP2D6 Interindividual Variability in Patients Under Pharmacological Treatments
    De Gregori, Manuela
    Allegri, Massimo
    De Gregori, Simona
    Garbin, Giulia
    Tinelli, Carmine
    Regazzi, Mario
    Govoni, Stefano
    Ranzani, Guglielmina Nadia
    CURRENT DRUG METABOLISM, 2010, 11 (03) : 276 - 282
  • [23] THE EFFECT OF SELECTIVE SEROTONIN REUPTAKE INHIBITORS ON CYTOCHROME-P4502D6 (CYP2D6) ACTIVITY IN HUMAN LIVER-MICROSOMES
    CREWE, HK
    LENNARD, MS
    TUCKER, GT
    WOODS, FR
    HADDOCK, RE
    BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1992, 34 (03) : 262 - 265
  • [24] Metabolism of dexfenfluramine in human liver microsomes and by recombinant enzymes: role of CYP2D6 and 1A2
    Haritos, VS
    Ching, MS
    Ghabrial, H
    Gross, AS
    Taavitsainen, P
    Pelkonen, O
    Battaglia, SE
    Smallwood, RA
    Ahokas, JT
    PHARMACOGENETICS, 1998, 8 (05): : 423 - 432
  • [25] CYP2D6 Phenotyping Using Urine, Plasma, and Saliva Metabolic Ratios to Assess the Impact of CYP2D6*10 on Interindividual Variation in a Chinese Population
    Chen, Rui
    Zheng, Xin
    Hu, Pei
    FRONTIERS IN PHARMACOLOGY, 2017, 8
  • [26] Investigation of CYP3A4 and CYP2D6 Interactions of Withania somnifera and Centella asiatica in Human Liver Microsomes
    Savai, Jay
    Varghese, Alice
    Pandita, Nancy
    Chintamaneni, Meena
    PHYTOTHERAPY RESEARCH, 2015, 29 (05) : 785 - 790
  • [27] Genetic Variation in CYP2D6 and CYP2C8 is Associated With Differences in Human Brain Expression
    Giegerich, Mellissa
    Prettyman, Greer
    Ursini, Gianluca
    Shin, Joo Heon
    Jaffe, Andrew
    Hyde, Thomas M.
    Kleinman, Joel
    Weinberger, Daniel R.
    Bigos, Kristin
    NEUROPSYCHOPHARMACOLOGY, 2016, 41 : S550 - S550
  • [28] Interactions of amphetamine analogs with human liver CYP2D6
    Wu, DF
    Otton, SV
    Inaba, T
    Kalow, W
    Sellers, EM
    BIOCHEMICAL PHARMACOLOGY, 1997, 53 (11) : 1605 - 1612
  • [29] GENETIC POLYMORPHISM IN CYTOCHROME P450 2D6 (CYP2D6): POPULATION DISTRIBUTION OF CYP2D6 ACTIVITY
    Neafsey, Patricia
    Ginsberg, Gary
    Hattis, Dale
    Sonawane, Babasaheb
    JOURNAL OF TOXICOLOGY AND ENVIRONMENTAL HEALTH-PART B-CRITICAL REVIEWS, 2009, 12 (5-6): : 334 - 361
  • [30] Developmental changes in human liver CYP2D6 expression
    Stevens, Jeffrey C.
    Marsh, Sandra A.
    Zaya, Matthew J.
    Regina, Karen J.
    Divakaran, Karthika
    Le, Min
    Hines, Ronald N.
    DRUG METABOLISM AND DISPOSITION, 2008, 36 (08) : 1587 - 1593