Structure-Activity Relationships of the Peptide Kappa Opioid Receptor Antagonist Zyklophin

被引:0
|
作者
Joshi, A. A. [1 ]
Murray, T. F. [2 ]
Aldrich, J. V. [1 ]
机构
[1] Univ Kansas, Dept Med Chem, Lawrence, KS 66045 USA
[2] Creighton Univ, Sch Med, Dept Pharmacol, Omaha, NE 68178 USA
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:477 / 477
页数:1
相关论文
共 50 条
  • [21] THE CRYSTAL-STRUCTURE OF A BIMORPHINAN WITH HIGHLY SELECTIVE KAPPA-OPIOID RECEPTOR ANTAGONIST ACTIVITY
    URBANCZYKLIPKOWSKA, Z
    ETTER, MC
    LIPKOWSKI, AW
    PORTOGHESE, PS
    JOURNAL OF MOLECULAR STRUCTURE, 1987, 159 (3-4) : 287 - 295
  • [22] BUPRENORPHINE HAS POTENT KAPPA-OPIOID RECEPTOR ANTAGONIST ACTIVITY
    LEANDER, JD
    NEUROPHARMACOLOGY, 1987, 26 (09) : 1445 - 1447
  • [23] Structure-activity relationships of a potent and selective Ca2+ Receptor antagonist.
    Callahan, JF
    Barton, L
    Bryan, WM
    Burgess, JL
    DelMar, R
    Fox, J
    Gleason, JG
    Gorycki, P
    Gowen, M
    Huffman, WF
    Lago, AM
    Nemeth, E
    Nguyen, TT
    Smith, BR
    Stroup, G
    Bhatnagar, PK
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 221 : U35 - U35
  • [24] Structure-Activity Relationships of [des-Arg7]Dynorphin A Analogues at the κ Opioid Receptor
    Ramos-Colon, Cyf N.
    Lee, Yeon Sun
    Remesic, Michael
    Hall, Sara M.
    LaVigne, Justin
    Davis, Peg
    Sandweiss, Alexander J.
    McIntosh, Mary I.
    Hanson, Jessica
    Largent-Milnes, Tally M.
    Vanderah, Todd W.
    Streicher, John
    Porreca, Frank
    Hruby, Victor J.
    JOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (22) : 10291 - 10298
  • [25] 3D quantitative and qualitative structure-activity relationships of the δ-opioid receptor antagonists
    Chun, Sun
    Lee, Jee-Young
    Ro, Seong-Gu
    Jeong, Ki-Woong
    Kim, Yangmee
    Yoon, Chang-Ju
    Bulletin of the Korean Chemical Society, 2008, 29 (03) : 656 - 662
  • [26] 3D quantitative and qualitative structure-activity relationships of the δ-opioid receptor antagonists
    Chun, Sun
    Lee, Jee-Young
    Ro, Seong-Gu
    Jeong, Ki-Woong
    Kim, Yangmee
    Yoon, Chang-Ju
    BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2008, 29 (03): : 656 - 662
  • [27] TENA, A SELECTIVE KAPPA OPIOID RECEPTOR ANTAGONIST
    PORTOGHESE, PS
    TAKEMORI, AE
    LIFE SCIENCES, 1985, 36 (08) : 801 - 805
  • [28] BUPRENORPHINE IS AN ANTAGONIST AT THE KAPPA-OPIOID RECEPTOR
    RICHARDS, ML
    SADEE, W
    PHARMACEUTICAL RESEARCH, 1985, (04) : 178 - 181
  • [29] A Structure-Activity Relationship Comparison of Imidazodiazepines Binding at Kappa, Mu, and Delta Opioid Receptors and the GABAA Receptor
    Li, Guanguan
    Nieman, Amanda N.
    Mian, Md Yeunus
    Zahn, Nicolas M.
    Mikulsky, Brandon N.
    Poe, Michael M.
    Methuku, Kashi R.
    Liu, Yongfeng
    Cook, James M.
    Stafford, Douglas C.
    Arnold, Leggy A.
    MOLECULES, 2020, 25 (17):
  • [30] A Bicyclic Analog of the Linear Peptide Arodyn Is a Potent and Selective Kappa Opioid Receptor Antagonist
    Gisemba, Solomon A.
    Ferracane, Michael J.
    Murray, Thomas F.
    Aldrich, Jane V.
    MOLECULES, 2024, 29 (13):