Synthesis of substituted 3-trifluoromethylbenzo[b]thiophenes

被引：21
|
作者：
Owton, WM [1 ]
机构：
[1] Eli Lilly & Co, Lilly Res Ctr Ltd, Windlesham GU20 6PH, Surrey, England
来源：
TETRAHEDRON LETTERS | 2003年 / 44卷 / 38期
关键词：
lithiation; trifluoromethylbenzothiophenes;
D O I：
10.1016/S0040-4039(03)01811-2
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A straightforward method for the synthesis of 5/6-substituted 3-trifluoromethylbenzo[b]thiophenes and their precursor o-fluorinated trifluoro acetophenones is reported. (C) 2003 Elsevier Ltd. All rights reserved.
引用
收藏
页码：7147 / 7149
页数：3
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